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Development of covalent chemogenetic K2P channel activators.
Deal, Parker E; Lee, Haerim; Mondal, Abhisek; Lolicato, Marco; Mendonça, Philipe Ribeiro Furtado de; Black, Holly; Jang, Seil; El-Hilali, Xochina; Bryant, Clifford; Isacoff, Ehud Y; Renslo, Adam R; Minor, Daniel L.
Affiliation
  • Deal PE; Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA 93858-2330, USA; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA 93858-2330, USA.
  • Lee H; Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA 93858-2330, USA.
  • Mondal A; Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA 93858-2330, USA.
  • Lolicato M; Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA 93858-2330, USA.
  • Mendonça PRF; Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, CA 94720, USA.
  • Black H; Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, CA 94720, USA.
  • Jang S; Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA 93858-2330, USA.
  • El-Hilali X; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA 93858-2330, USA.
  • Bryant C; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA 93858-2330, USA.
  • Isacoff EY; Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, CA 94720, USA; Helen Wills Neuroscience Institute, University of California, Berkeley, Berkeley, CA 94720, USA; Weill Neurohub, University of California, Berkeley, Berkeley, CA 94720, USA; Molecular Biophysics an
  • Renslo AR; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA 93858-2330, USA. Electronic address: adam.renslo@ucsf.edu.
  • Minor DL; Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA 93858-2330, USA; Molecular Biophysics and Integrated Bio-imaging Division, Lawrence Berkeley National Laboratory, Berkeley, CA 94720 USA; Departments of Biochemistry and Biophysics, and Cellular and Molecul
Cell Chem Biol ; 31(7): 1305-1323.e9, 2024 Jul 18.
Article in En | MEDLINE | ID: mdl-39029456

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Potassium Channels, Tandem Pore Domain Limits: Animals / Humans Language: En Journal: Cell Chem Biol Year: 2024 Document type: Article Affiliation country: Estados Unidos Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Potassium Channels, Tandem Pore Domain Limits: Animals / Humans Language: En Journal: Cell Chem Biol Year: 2024 Document type: Article Affiliation country: Estados Unidos Country of publication: Estados Unidos