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Selective estrogen receptor modulators with conformationally restricted side chains. Synthesis and structure-activity relationship of ERalpha-selective tetrahydroisoquinoline ligands.
Renaud, Johanne; Bischoff, Serge François; Buhl, Thomas; Floersheim, Philipp; Fournier, Brigitte; Geiser, Martin; Halleux, Christine; Kallen, Joerg; Keller, Hansjoerg; Ramage, Paul.
Affiliation
  • Renaud J; Novartis Institute for Biomedical Research, WKL-136.6.81, CH-4002 Basel, Switzerland. johanne.renaud@pharma.novartis.com
J Med Chem ; 48(2): 364-79, 2005 Jan 27.
Article in En | MEDLINE | ID: mdl-15658851
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Collection: 01-internacional Database: MEDLINE Main subject: Selective Estrogen Receptor Modulators / Tetrahydroisoquinolines / Estrogen Receptor alpha / Isoquinolines Limits: Animals / Female / Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2005 Document type: Article Affiliation country: Switzerland Country of publication: United States
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Collection: 01-internacional Database: MEDLINE Main subject: Selective Estrogen Receptor Modulators / Tetrahydroisoquinolines / Estrogen Receptor alpha / Isoquinolines Limits: Animals / Female / Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2005 Document type: Article Affiliation country: Switzerland Country of publication: United States