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[N-methyl-3H3]AZ10419369 binding to the 5-HT1B receptor: in vitro characterization and in vivo receptor occupancy.
Maier, Donna L; Sobotka-Briner, Cindy; Ding, Min; Powell, Mark E; Jiang, Qiaoling; Hill, Geraldine; Heys, J Richard; Elmore, Charles S; Pierson, M Edward; Mrzljak, Ladislav.
Affiliation
  • Maier DL; Department of Neuroscience, AstraZeneca, Research Center, B1119A, 1800 Concord Pike, Wilmington, DE 19850, USA. donna.maier@astrazeneca.com
J Pharmacol Exp Ther ; 330(1): 342-51, 2009 Jul.
Article in En | MEDLINE | ID: mdl-19401496

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperazines / Serotonin Antagonists / Tritium / Benzopyrans / Morpholines / Radiopharmaceuticals / Receptor, Serotonin, 5-HT1B / Serotonin 5-HT1 Receptor Antagonists Limits: Animals / Humans / Male Language: En Journal: J Pharmacol Exp Ther Year: 2009 Document type: Article Affiliation country: United States Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperazines / Serotonin Antagonists / Tritium / Benzopyrans / Morpholines / Radiopharmaceuticals / Receptor, Serotonin, 5-HT1B / Serotonin 5-HT1 Receptor Antagonists Limits: Animals / Humans / Male Language: En Journal: J Pharmacol Exp Ther Year: 2009 Document type: Article Affiliation country: United States Country of publication: United States