Peptidyl succinimidyl peptides as taspase 1 inhibitors.

van den Boom, Johannes; Mamic, Marija; Baccelliere, Daniele; Zweerink, Susanne; Kaschani, Farnusch; Knauer, Shirley; Bayer, Peter; Kaiser, Markus

van den Boom, Johannes; Mamic, Marija; Baccelliere, Daniele; Zweerink, Susanne; Kaschani, Farnusch; Knauer, Shirley; Bayer, Peter; Kaiser, Markus.

Affiliation

van den Boom J; Strukturelle Biochemie, Universität Duisburg-Essen, Zentrum für Medizinische Biotechnologie, Universitätsstrasse 2, 45117 Essen (Germany).

Chembiochem ; 15(15): 2233-7, 2014 Oct 13.

Article in En | MEDLINE | ID: mdl-25146997

Subject(s)

Endopeptidases/metabolism; Peptides/pharmacology; Protease Inhibitors/pharmacology; Dose-Response Relationship, Drug; Humans; Molecular Conformation; Peptides/chemical synthesis; Peptides/chemistry; Protease Inhibitors/chemical synthesis; Protease Inhibitors/chemistry; Structure-Activity Relationship

Key words

Taspase; activity-based profiling; cancer; inhibitors; mechanism-based design; protease

Fulltext

Add to My VHL

XML

PubMed Links

Search on Google

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Endopeptidases / Peptides / Protease Inhibitors Limits: Humans Language: En Journal: Chembiochem Journal subject: BIOQUIMICA Year: 2014 Document type: Article Country of publication: Germany

Fulltext

Add to My VHL

XML

PubMed Links

Search on Google