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Targeting methionyl tRNA synthetase: design, synthesis and antibacterial activity against Clostridium difficile of novel 3-biaryl-N-benzylpropan-1-amine derivatives.
Eissa, Ahmed G; Blaxland, James A; Williams, Rhodri O; Metwally, Kamel A; El-Adl, Sobhy M; Lashine, El-Sayed M; Baillie, Leslie W J; Simons, Claire.
Affiliation
  • Eissa AG; a School of Pharmacy & Pharmaceutical Sciences, Cardiff University , King Edward VII Avenue, Cardiff, Wales , UK and.
  • Blaxland JA; b Department of Medicinal Chemistry , Faculty of Pharmacy, Zagazig University , Zagazig , Egypt.
  • Williams RO; a School of Pharmacy & Pharmaceutical Sciences, Cardiff University , King Edward VII Avenue, Cardiff, Wales , UK and.
  • Metwally KA; a School of Pharmacy & Pharmaceutical Sciences, Cardiff University , King Edward VII Avenue, Cardiff, Wales , UK and.
  • El-Adl SM; b Department of Medicinal Chemistry , Faculty of Pharmacy, Zagazig University , Zagazig , Egypt.
  • Lashine el-SM; b Department of Medicinal Chemistry , Faculty of Pharmacy, Zagazig University , Zagazig , Egypt.
  • Baillie LW; b Department of Medicinal Chemistry , Faculty of Pharmacy, Zagazig University , Zagazig , Egypt.
  • Simons C; a School of Pharmacy & Pharmaceutical Sciences, Cardiff University , King Edward VII Avenue, Cardiff, Wales , UK and.
J Enzyme Inhib Med Chem ; 31(6): 1694-7, 2016 Dec.
Article in En | MEDLINE | ID: mdl-26899668

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Propane / Clostridioides difficile / Methionine-tRNA Ligase / Anti-Bacterial Agents Language: En Journal: J Enzyme Inhib Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2016 Document type: Article Country of publication: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Propane / Clostridioides difficile / Methionine-tRNA Ligase / Anti-Bacterial Agents Language: En Journal: J Enzyme Inhib Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2016 Document type: Article Country of publication: United kingdom