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Identification and biological activity of 6-alkyl-substituted 3-methyl-pyridine-2-carbonyl amino dimethyl-benzoic acid EP4 antagonists.
Blanco, Maria-Jesus; Vetman, Tatiana; Chandrasekhar, Srinivasan; Fisher, Matthew J; Harvey, Anita; Kuklish, Steven L; Chambers, Mark; Lin, Chaohua; Mudra, Daniel; Oskins, Jennifer; Wang, Xu-Shan; Yu, Xiao-Peng; Warshawsky, Alan M.
Affiliation
  • Blanco MJ; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States. Electronic address: blanco_maria@lilly.com.
  • Vetman T; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Chandrasekhar S; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Fisher MJ; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Harvey A; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Kuklish SL; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Chambers M; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Lin C; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Mudra D; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Oskins J; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Wang XS; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Yu XP; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
  • Warshawsky AM; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN 46285, United States.
Bioorg Med Chem Lett ; 26(9): 2303-7, 2016 May 01.
Article in En | MEDLINE | ID: mdl-27020304

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Benzoates / Receptors, Prostaglandin E, EP4 Subtype Type of study: Diagnostic_studies Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2016 Document type: Article Country of publication: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Benzoates / Receptors, Prostaglandin E, EP4 Subtype Type of study: Diagnostic_studies Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2016 Document type: Article Country of publication: United kingdom