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Inhibition of cytochrome P450 enzymes by saturated and unsaturated fatty acids in human liver microsomes, characterization of enzyme kinetics in the presence of bovine serum albumin (0.1 and 1.0% w/v) and in vitro - in vivo extrapolation of hepatic clearance.
Palacharla, Raghava Choudary; Uthukam, Venkatesham; Manoharan, Arunkumar; Ponnamaneni, Ranjith Kumar; Padala, Nagasurya Prakash; Boggavarapu, Rajesh Kumar; Bhyrapuneni, Gopinadh; Ajjala, Devender Reddy; Nirogi, Ramakrishna.
Affiliation
  • Palacharla RC; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd, Jeedimetla, Hyderabad, India.
  • Uthukam V; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd, Jeedimetla, Hyderabad, India.
  • Manoharan A; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd, Jeedimetla, Hyderabad, India.
  • Ponnamaneni RK; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd, Jeedimetla, Hyderabad, India.
  • Padala NP; Biopharmaceutical Research, Suven Life Sciences Ltd, Pashamylaram, Medak, India.
  • Boggavarapu RK; Biopharmaceutical Research, Suven Life Sciences Ltd, Pashamylaram, Medak, India.
  • Bhyrapuneni G; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd, Jeedimetla, Hyderabad, India.
  • Ajjala DR; Biopharmaceutical Research, Suven Life Sciences Ltd, Pashamylaram, Medak, India.
  • Nirogi R; Discovery Research, Suven Life Sciences Ltd, Banjara Hills, Hyderabad, India. Electronic address: nvsrk@suven.com.
Eur J Pharm Sci ; 101: 80-89, 2017 Apr 01.
Article in En | MEDLINE | ID: mdl-28179134

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Serum Albumin, Bovine / Microsomes, Liver / Cytochrome P-450 Enzyme System / Fatty Acids / Fatty Acids, Unsaturated / Cytochrome P-450 Enzyme Inhibitors / Liver Type of study: Prognostic_studies Limits: Humans Language: En Journal: Eur J Pharm Sci Journal subject: FARMACIA / FARMACOLOGIA / QUIMICA Year: 2017 Document type: Article Affiliation country: India Country of publication: Netherlands

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Serum Albumin, Bovine / Microsomes, Liver / Cytochrome P-450 Enzyme System / Fatty Acids / Fatty Acids, Unsaturated / Cytochrome P-450 Enzyme Inhibitors / Liver Type of study: Prognostic_studies Limits: Humans Language: En Journal: Eur J Pharm Sci Journal subject: FARMACIA / FARMACOLOGIA / QUIMICA Year: 2017 Document type: Article Affiliation country: India Country of publication: Netherlands