Inhibition of cytochrome P450 enzymes by saturated and unsaturated fatty acids in human liver microsomes, characterization of enzyme kinetics in the presence of bovine serum albumin (0.1 and 1.0% w/v) and in vitro - in vivo extrapolation of hepatic clearance.
Eur J Pharm Sci
; 101: 80-89, 2017 Apr 01.
Article
in En
| MEDLINE
| ID: mdl-28179134
Key words
Full text:
1
Collection:
01-internacional
Database:
MEDLINE
Main subject:
Serum Albumin, Bovine
/
Microsomes, Liver
/
Cytochrome P-450 Enzyme System
/
Fatty Acids
/
Fatty Acids, Unsaturated
/
Cytochrome P-450 Enzyme Inhibitors
/
Liver
Type of study:
Prognostic_studies
Limits:
Humans
Language:
En
Journal:
Eur J Pharm Sci
Journal subject:
FARMACIA
/
FARMACOLOGIA
/
QUIMICA
Year:
2017
Document type:
Article
Affiliation country:
India
Country of publication:
Netherlands