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Targeting S-adenosylmethionine biosynthesis with a novel allosteric inhibitor of Mat2A.
Quinlan, Casey L; Kaiser, Stephen E; Bolaños, Ben; Nowlin, Dawn; Grantner, Rita; Karlicek-Bryant, Shannon; Feng, Jun Li; Jenkinson, Stephen; Freeman-Cook, Kevin; Dann, Stephen G; Wang, Xiaoli; Wells, Peter A; Fantin, Valeria R; Stewart, Al E; Grant, Stephan K.
Affiliation
  • Quinlan CL; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
  • Kaiser SE; Oncology Medicinal Chemistry, Pfizer Inc., San Diego, California, USA.
  • Bolaños B; Oncology Medicinal Chemistry, Pfizer Inc., San Diego, California, USA.
  • Nowlin D; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
  • Grantner R; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
  • Karlicek-Bryant S; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
  • Feng JL; Oncology Medicinal Chemistry, Pfizer Inc., San Diego, California, USA.
  • Jenkinson S; Drug Safety and Pharmacology, Pfizer Inc., San Diego, California, USA.
  • Freeman-Cook K; Oncology Medicinal Chemistry, Pfizer Inc., San Diego, California, USA.
  • Dann SG; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
  • Wang X; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
  • Wells PA; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
  • Fantin VR; ORIC Pharmaceuticals, South San Francisco, California, USA.
  • Stewart AE; Oncology Medicinal Chemistry, Pfizer Inc., San Diego, California, USA.
  • Grant SK; Oncology Research and Development, Pfizer Inc., San Diego, California, USA.
Nat Chem Biol ; 13(7): 785-792, 2017 Jul.
Article in En | MEDLINE | ID: mdl-28553945

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / S-Adenosylmethionine / Triazoles / Methionine Adenosyltransferase Limits: Humans Language: En Journal: Nat Chem Biol Journal subject: BIOLOGIA / QUIMICA Year: 2017 Document type: Article Affiliation country: United States Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / S-Adenosylmethionine / Triazoles / Methionine Adenosyltransferase Limits: Humans Language: En Journal: Nat Chem Biol Journal subject: BIOLOGIA / QUIMICA Year: 2017 Document type: Article Affiliation country: United States Country of publication: United States