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Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a Gαi/o protein inhibitor.
Porcu, Alessandra; Melis, Miriam; Turecek, Rostislav; Ullrich, Celine; Mocci, Ignazia; Bettler, Bernhard; Gessa, Gian Luigi; Castelli, M Paola.
Affiliation
  • Porcu A; Department of Biomedical Sciences, University of Cagliari, 09042, Monserrato, Italy; Department of Biomedicine, University of Basel, Klingelbergstrasse 50-70, CH-4056, Basel, Switzerland.
  • Melis M; Department of Biomedical Sciences, University of Cagliari, 09042, Monserrato, Italy.
  • Turecek R; Department of Biomedicine, University of Basel, Klingelbergstrasse 50-70, CH-4056, Basel, Switzerland.
  • Ullrich C; Department of Biomedicine, University of Basel, Klingelbergstrasse 50-70, CH-4056, Basel, Switzerland.
  • Mocci I; Institute of Translational Pharmacology, National Research Council of Italy (CNR) U.O.S. of Cagliari, 09010, Pula, Italy.
  • Bettler B; Department of Biomedicine, University of Basel, Klingelbergstrasse 50-70, CH-4056, Basel, Switzerland.
  • Gessa GL; Department of Biomedical Sciences, University of Cagliari, 09042, Monserrato, Italy; Guy Everett Laboratory, University of Cagliari, 09042, Monserrato, Italy; Neuroscience Institute, National Research Council of Italy (CNR), Cagliari, Italy; Center of Excellence "Neurobiology of Addiction", Universi
  • Castelli MP; Department of Biomedical Sciences, University of Cagliari, 09042, Monserrato, Italy; Center of Excellence "Neurobiology of Addiction", University of Cagliari, 09042, Monserrato, Italy. Electronic address: castelli@unica.it.
Neuropharmacology ; 133: 107-120, 2018 05 01.
Article in En | MEDLINE | ID: mdl-29407764

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Pyrazoles / GTP-Binding Protein alpha Subunits, Gi-Go / Receptor, Cannabinoid, CB1 / Cannabinoid Receptor Antagonists Limits: Animals / Humans Language: En Journal: Neuropharmacology Year: 2018 Document type: Article Affiliation country: Switzerland

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Pyrazoles / GTP-Binding Protein alpha Subunits, Gi-Go / Receptor, Cannabinoid, CB1 / Cannabinoid Receptor Antagonists Limits: Animals / Humans Language: En Journal: Neuropharmacology Year: 2018 Document type: Article Affiliation country: Switzerland