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Bioinspired co-crystals of Imatinib providing enhanced kinetic solubility.
Reggane, Maude; Wiest, Johannes; Saedtler, Marco; Harlacher, Cornelius; Gutmann, Marcus; Zottnick, Sven H; Piechon, Philippe; Dix, Ina; Müller-Buschbaum, Klaus; Holzgrabe, Ulrike; Meinel, Lorenz; Galli, Bruno.
Affiliation
  • Reggane M; Novartis Pharma AG, Novartis Campus, CH-4056 Basel, Switzerland.
  • Wiest J; Institute for Pharmacy and Food Chemistry, University of Wuerzburg, Am Hubland, DE-97074 Wuerzburg, Germany.
  • Saedtler M; Institute for Pharmacy and Food Chemistry, University of Wuerzburg, Am Hubland, DE-97074 Wuerzburg, Germany.
  • Harlacher C; Novartis Pharma AG, Novartis Campus, CH-4056 Basel, Switzerland.
  • Gutmann M; Institute for Pharmacy and Food Chemistry, University of Wuerzburg, Am Hubland, DE-97074 Wuerzburg, Germany.
  • Zottnick SH; Institute for Inorganic Chemistry, University of Wuerzburg, Am Hubland, DE-97074 Wuerzburg, Germany.
  • Piechon P; Novartis Pharma AG, Novartis Campus, CH-4056 Basel, Switzerland.
  • Dix I; Novartis Pharma AG, Novartis Campus, CH-4056 Basel, Switzerland.
  • Müller-Buschbaum K; Institute for Inorganic Chemistry, University of Wuerzburg, Am Hubland, DE-97074 Wuerzburg, Germany.
  • Holzgrabe U; Institute for Pharmacy and Food Chemistry, University of Wuerzburg, Am Hubland, DE-97074 Wuerzburg, Germany.
  • Meinel L; Institute for Pharmacy and Food Chemistry, University of Wuerzburg, Am Hubland, DE-97074 Wuerzburg, Germany. Electronic address: Lorenz.meinel@uni-wuerzburg.de.
  • Galli B; Novartis Pharma AG, Novartis Campus, CH-4056 Basel, Switzerland.
Eur J Pharm Biopharm ; 128: 290-299, 2018 Jul.
Article in En | MEDLINE | ID: mdl-29733951

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Drug Liberation / Imatinib Mesylate / Gallic Acid Language: En Journal: Eur J Pharm Biopharm Journal subject: FARMACIA / FARMACOLOGIA Year: 2018 Document type: Article Affiliation country: Switzerland

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Drug Liberation / Imatinib Mesylate / Gallic Acid Language: En Journal: Eur J Pharm Biopharm Journal subject: FARMACIA / FARMACOLOGIA Year: 2018 Document type: Article Affiliation country: Switzerland