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Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position.
Felicetti, Tommaso; Cannalire, Rolando; Nizi, Maria Giulia; Tabarrini, Oriana; Massari, Serena; Barreca, Maria Letizia; Manfroni, Giuseppe; Schindler, Bryan D; Cecchetti, Violetta; Kaatz, Glenn W; Sabatini, Stefano.
Affiliation
  • Felicetti T; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Cannalire R; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Nizi MG; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Tabarrini O; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Massari S; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Barreca ML; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Manfroni G; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Schindler BD; John D. Dingell Department of Veterans Affairs Medical Centre, Division of Infectious Diseases, School of Medicine, Wayne State University, Detroit, MI 48201, United States.
  • Cecchetti V; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy.
  • Kaatz GW; John D. Dingell Department of Veterans Affairs Medical Centre, Division of Infectious Diseases, School of Medicine, Wayne State University, Detroit, MI 48201, United States; Department of Internal Medicine, Division of Infectious Diseases, School of Medicine, Wayne State University, Detroit, MI 4820
  • Sabatini S; Department of Pharmaceutical Sciences, University of Perugia, via del Liceo 1, 06123, Perugia, Italy. Electronic address: stefano.sabatini@unipg.it.
Eur J Med Chem ; 155: 428-433, 2018 Jul 15.
Article in En | MEDLINE | ID: mdl-29908437

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / Staphylococcus aureus / Bacterial Proteins / Multidrug Resistance-Associated Proteins / Anti-Bacterial Agents Limits: Humans Language: En Journal: Eur J Med Chem Year: 2018 Document type: Article Affiliation country: Italy Country of publication: France

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / Staphylococcus aureus / Bacterial Proteins / Multidrug Resistance-Associated Proteins / Anti-Bacterial Agents Limits: Humans Language: En Journal: Eur J Med Chem Year: 2018 Document type: Article Affiliation country: Italy Country of publication: France