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Identification of potent RORß modulators: Scaffold variation.
Doebelin, Christelle; Patouret, Rémi; Garcia-Ordonez, Ruben D; Chang, Mi Ra; Dharmarajan, Venkatasubramanian; Novick, Scott; Ciesla, Anthony; Campbell, Sean; Solt, Laura A; Griffin, Patrick R; Kamenecka, Theodore M.
Affiliation
  • Doebelin C; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Patouret R; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Garcia-Ordonez RD; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Chang MR; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Dharmarajan V; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Novick S; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Ciesla A; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Campbell S; The Scripps Research Institute, Scripps Florida, Department of Immunology and Microbiology, 130 Scripps Way #C2A, Jupiter, FL 33458, USA.
  • Solt LA; The Scripps Research Institute, Scripps Florida, Department of Immunology and Microbiology, 130 Scripps Way #C2A, Jupiter, FL 33458, USA.
  • Griffin PR; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA.
  • Kamenecka TM; The Scripps Research Institute, Scripps Florida, Department of Molecular Medicine, 130 Scripps Way #A2A, Jupiter, FL 33458, USA. Electronic address: kameneck@scripps.edu.
Bioorg Med Chem Lett ; 28(19): 3210-3215, 2018 10 15.
Article in En | MEDLINE | ID: mdl-30143422

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Thiophenes / Nuclear Receptor Subfamily 1, Group F, Member 2 Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2018 Document type: Article Affiliation country: United States Country of publication: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Thiophenes / Nuclear Receptor Subfamily 1, Group F, Member 2 Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2018 Document type: Article Affiliation country: United States Country of publication: United kingdom