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Halogen-substituted anthranilic acid derivatives provide a novel chemical platform for androgen receptor antagonists.
Roell, Daniela; Rösler, Thomas W; Hessenkemper, Wiebke; Kraft, Florian; Hauschild, Monique; Bartsch, Sophie; Abraham, Tsion E; Houtsmuller, Adriaan B; Matusch, Rudolf; van Royen, Martin E; Baniahmad, Aria.
Affiliation
  • Roell D; Institute of Human Genetics, Jena University Hospital, Jena, Germany; Center for Sepsis Control and Care (CSCC), Jena University Hospital, Jena, Germany.
  • Rösler TW; Institute of Pharmaceutical Chemistry, Philipps-University, Marburg, Germany.
  • Hessenkemper W; Institute of Human Genetics, Jena University Hospital, Jena, Germany.
  • Kraft F; Institute of Human Genetics, Jena University Hospital, Jena, Germany.
  • Hauschild M; Institute of Human Genetics, Jena University Hospital, Jena, Germany.
  • Bartsch S; Institute of Human Genetics, Jena University Hospital, Jena, Germany.
  • Abraham TE; Department of Pathology and Erasmus Optical Imaging Center OIC, Erasmus MC, Rotterdam, the Netherlands.
  • Houtsmuller AB; Department of Pathology and Erasmus Optical Imaging Center OIC, Erasmus MC, Rotterdam, the Netherlands.
  • Matusch R; Institute of Pharmaceutical Chemistry, Philipps-University, Marburg, Germany.
  • van Royen ME; Department of Pathology and Erasmus Optical Imaging Center OIC, Erasmus MC, Rotterdam, the Netherlands.
  • Baniahmad A; Institute of Human Genetics, Jena University Hospital, Jena, Germany. Electronic address: aria.baniahmad@med.uni-jena.de.
J Steroid Biochem Mol Biol ; 188: 59-70, 2019 04.
Article in En | MEDLINE | ID: mdl-30615932

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Androgen Receptor Antagonists / Ortho-Aminobenzoates Type of study: Prognostic_studies Limits: Animals / Humans / Male Language: En Journal: J Steroid Biochem Mol Biol Journal subject: BIOLOGIA MOLECULAR / BIOQUIMICA Year: 2019 Document type: Article Affiliation country: Germany Country of publication: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Androgen Receptor Antagonists / Ortho-Aminobenzoates Type of study: Prognostic_studies Limits: Animals / Humans / Male Language: En Journal: J Steroid Biochem Mol Biol Journal subject: BIOLOGIA MOLECULAR / BIOQUIMICA Year: 2019 Document type: Article Affiliation country: Germany Country of publication: United kingdom