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A chemical toolbox for the study of bromodomains and epigenetic signaling.
Wu, Qin; Heidenreich, David; Zhou, Stanley; Ackloo, Suzanne; Krämer, Andreas; Nakka, Kiran; Lima-Fernandes, Evelyne; Deblois, Genevieve; Duan, Shili; Vellanki, Ravi N; Li, Fengling; Vedadi, Masoud; Dilworth, Jeffrey; Lupien, Mathieu; Brennan, Paul E; Arrowsmith, Cheryl H; Müller, Susanne; Fedorov, Oleg; Filippakopoulos, Panagis; Knapp, Stefan.
Affiliation
  • Wu Q; Structural Genomics Consortium, University of Toronto, Toronto, ON, M5G 1L7, Canada.
  • Heidenreich D; Princess Margaret Cancer Centre, University Health Network, Toronto, M5G 2M9, ON, Canada.
  • Zhou S; Department of Medical Biophysics, University of Toronto, Toronto, M5G 2M9, ON, Canada.
  • Ackloo S; Structural Genomics Consortium, University of Toronto, Toronto, ON, M5G 1L7, Canada.
  • Krämer A; Structural Genomics Consortium, Buchmann Institute for Life Sciences, Goethe-University Frankfurt, 60438, Frankfurt, Germany.
  • Nakka K; Princess Margaret Cancer Centre, University Health Network, Toronto, M5G 2M9, ON, Canada.
  • Lima-Fernandes E; Department of Medical Biophysics, University of Toronto, Toronto, M5G 2M9, ON, Canada.
  • Deblois G; Structural Genomics Consortium, University of Toronto, Toronto, ON, M5G 1L7, Canada.
  • Duan S; Structural Genomics Consortium, Buchmann Institute for Life Sciences, Goethe-University Frankfurt, 60438, Frankfurt, Germany.
  • Vellanki RN; Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt, 60438, Frankfurt, Germany.
  • Li F; Sprott Centre for Stem Cell Research, Regenerative Medicine Program, Ottawa Hospital Research Institute, Ottawa, K1H 8L6, ON, Canada.
  • Vedadi M; Structural Genomics Consortium, University of Toronto, Toronto, ON, M5G 1L7, Canada.
  • Dilworth J; Princess Margaret Cancer Centre, University Health Network, Toronto, M5G 2M9, ON, Canada.
  • Lupien M; Department of Medical Biophysics, University of Toronto, Toronto, M5G 2M9, ON, Canada.
  • Brennan PE; Princess Margaret Cancer Centre, University Health Network, Toronto, M5G 2M9, ON, Canada.
  • Arrowsmith CH; Department of Medical Biophysics, University of Toronto, Toronto, M5G 2M9, ON, Canada.
  • Müller S; Princess Margaret Cancer Centre, University Health Network, Toronto, M5G 2M9, ON, Canada.
  • Fedorov O; Department of Medical Biophysics, University of Toronto, Toronto, M5G 2M9, ON, Canada.
  • Filippakopoulos P; Princess Margaret Cancer Centre, University Health Network, Toronto, M5G 2M9, ON, Canada.
  • Knapp S; Structural Genomics Consortium, University of Toronto, Toronto, ON, M5G 1L7, Canada.
Nat Commun ; 10(1): 1915, 2019 04 23.
Article in En | MEDLINE | ID: mdl-31015424

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Gene Expression Regulation, Neoplastic / Protein Processing, Post-Translational / Epithelial Cells / Small Molecule Libraries / Antineoplastic Agents Limits: Humans Language: En Journal: Nat Commun Journal subject: BIOLOGIA / CIENCIA Year: 2019 Document type: Article Affiliation country: Canada Country of publication: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Gene Expression Regulation, Neoplastic / Protein Processing, Post-Translational / Epithelial Cells / Small Molecule Libraries / Antineoplastic Agents Limits: Humans Language: En Journal: Nat Commun Journal subject: BIOLOGIA / CIENCIA Year: 2019 Document type: Article Affiliation country: Canada Country of publication: United kingdom