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A practical synthesis of a novel DPAGT1 inhibitor, aminouridyl phenoxypiperidinbenzyl butanamide (APPB) for in vivo studies.
Mitachi, Katsuhiko; Kurosu, Shou M; Gillman, Cody D; Yun, Hyun Gi; Clemons, William M; Kurosu, Michio.
Affiliation
  • Mitachi K; Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Science Center, 881 Madison Avenue, Memphis, TN 38163, United States.
  • Kurosu SM; Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Science Center, 881 Madison Avenue, Memphis, TN 38163, United States.
  • Gillman CD; Division of Chemistry and Chemical Engineering, California Institute of Technology, 1200 E. California Blvd., Pasadena, CA 91125, United States.
  • Yun HG; Division of Chemistry and Chemical Engineering, California Institute of Technology, 1200 E. California Blvd., Pasadena, CA 91125, United States.
  • Clemons WM; Division of Chemistry and Chemical Engineering, California Institute of Technology, 1200 E. California Blvd., Pasadena, CA 91125, United States.
  • Kurosu M; Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Science Center, 881 Madison Avenue, Memphis, TN 38163, United States.
MethodsX ; 6: 2305-2321, 2019.
Article in En | MEDLINE | ID: mdl-31667130

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Guideline Language: En Journal: MethodsX Year: 2019 Document type: Article Affiliation country: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Guideline Language: En Journal: MethodsX Year: 2019 Document type: Article Affiliation country: United States