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Click chemistry-facilitated comprehensive identification of proteins adducted by antimicrobial 5-nitroimidazoles for discovery of alternative drug targets against giardiasis.
Lauwaet, Tineke; Miyamoto, Yukiko; Ihara, Sozaburo; Le, Christine; Kalisiak, Jaroslaw; Korthals, Keith A; Ghassemian, Majid; Smith, Diane K; Sharpless, K Barry; Fokin, Valery V; Eckmann, Lars.
Affiliation
  • Lauwaet T; Department of Pathology, University of California, San Diego, La Jolla, California, United States of America.
  • Miyamoto Y; Department of Medicine, University of California, San Diego, La Jolla, California, United States of America.
  • Ihara S; Department of Medicine, University of California, San Diego, La Jolla, California, United States of America.
  • Le C; Division of Gastroenterology, The Institute for Adult Diseases, Asahi Life Foundation, Tokyo, Japan.
  • Kalisiak J; Department of Medicine, University of California, San Diego, La Jolla, California, United States of America.
  • Korthals KA; Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, La Jolla, California, United States of America.
  • Ghassemian M; Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, La Jolla, California, United States of America.
  • Smith DK; Department of Chemistry and Biochemistry, University of California, San Diego, La Jolla, California, United States of America.
  • Sharpless KB; Department of Chemistry and Biochemistry, San Diego State University, San Diego, California, United States of America.
  • Fokin VV; Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, La Jolla, California, United States of America.
  • Eckmann L; Department of Chemistry, Dornsife College of Letters, Arts and Sciences, University of Southern California, Los Angeles, California, United States of America.
PLoS Negl Trop Dis ; 14(4): e0008224, 2020 04.
Article in En | MEDLINE | ID: mdl-32302296

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protozoan Proteins / Giardia lamblia / Drug Discovery / Click Chemistry / Indazoles / Antiparasitic Agents Type of study: Diagnostic_studies Limits: Animals Language: En Journal: PLoS Negl Trop Dis Journal subject: MEDICINA TROPICAL Year: 2020 Document type: Article Affiliation country: United States Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protozoan Proteins / Giardia lamblia / Drug Discovery / Click Chemistry / Indazoles / Antiparasitic Agents Type of study: Diagnostic_studies Limits: Animals Language: En Journal: PLoS Negl Trop Dis Journal subject: MEDICINA TROPICAL Year: 2020 Document type: Article Affiliation country: United States Country of publication: United States