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Identification of U83836E as a γ-glutamylcyclotransferase inhibitor that suppresses MCF7 breast cancer xenograft growth.
Ii, Hiromi; Nohara, Yukie; Yoshiya, Taku; Masuda, Shun; Tsuda, Shugo; Oishi, Shinya; Friedman, Jonathan; Kawabe, Takumi; Nakata, Susumu.
Affiliation
  • Ii H; Department of Clinical Oncology, Kyoto Pharmaceutical University, Misasagi-Nakauchicho 5, Yamashina, Kyoto, 607-8414, Japan.
  • Nohara Y; Peptide Institute, Inc., 7-2-9 Saito-Asagi, Ibaraki, Osaka, 567-0085, Japan.
  • Yoshiya T; Peptide Institute, Inc., 7-2-9 Saito-Asagi, Ibaraki, Osaka, 567-0085, Japan.
  • Masuda S; Peptide Institute, Inc., 7-2-9 Saito-Asagi, Ibaraki, Osaka, 567-0085, Japan.
  • Tsuda S; Peptide Institute, Inc., 7-2-9 Saito-Asagi, Ibaraki, Osaka, 567-0085, Japan.
  • Oishi S; Department of Medicinal Chemistry, Kyoto Pharmaceutical University, Yamashina-ku, Kyoto, 607-8412, Japan; Graduate School of Pharmaceutical Sciences, Kyoto University, Kyoto, 606-8501, Japan.
  • Friedman J; CanBas Co., Ltd., 2-2-1 Otemachi Numazu, Shizuoka, 410-0801, Japan.
  • Kawabe T; CanBas Co., Ltd., 2-2-1 Otemachi Numazu, Shizuoka, 410-0801, Japan.
  • Nakata S; Department of Clinical Oncology, Kyoto Pharmaceutical University, Misasagi-Nakauchicho 5, Yamashina, Kyoto, 607-8414, Japan. Electronic address: snakata@mb.kyoto-phu.ac.jp.
Biochem Biophys Res Commun ; 549: 128-134, 2021 04 16.
Article in En | MEDLINE | ID: mdl-33676180

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperazines / Breast Neoplasms / Chromans / Enzyme Inhibitors / Gamma-Glutamylcyclotransferase Type of study: Diagnostic_studies Limits: Animals / Female / Humans Language: En Journal: Biochem Biophys Res Commun Year: 2021 Document type: Article Affiliation country: Japan Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperazines / Breast Neoplasms / Chromans / Enzyme Inhibitors / Gamma-Glutamylcyclotransferase Type of study: Diagnostic_studies Limits: Animals / Female / Humans Language: En Journal: Biochem Biophys Res Commun Year: 2021 Document type: Article Affiliation country: Japan Country of publication: United States