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The synthetic varespladib molecule is a multi-functional inhibitor for PLA2 and PLA2-like ophidic toxins.
Salvador, Guilherme H M; Borges, Rafael J; Lomonte, Bruno; Lewin, Matthew R; Fontes, Marcos R M.
Affiliation
  • Salvador GHM; Departamento de Biofísica e Farmacologia, Instituto de Biociências, Universidade Estadual Paulista (UNESP), Botucatu, SP, Brazil.
  • Borges RJ; Departamento de Biofísica e Farmacologia, Instituto de Biociências, Universidade Estadual Paulista (UNESP), Botucatu, SP, Brazil.
  • Lomonte B; Instituto Clodomiro Picado, Facultad de Microbiología, Universidad de Costa Rica, San José, Costa Rica.
  • Lewin MR; Center for Exploration and Travel Health, California Academy of Sciences, San Francisco, CA 94118, USA.
  • Fontes MRM; Departamento de Biofísica e Farmacologia, Instituto de Biociências, Universidade Estadual Paulista (UNESP), Botucatu, SP, Brazil. Electronic address: marcos.fontes@unesp.br.
Biochim Biophys Acta Gen Subj ; 1865(7): 129913, 2021 07.
Article in En | MEDLINE | ID: mdl-33865953

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Bothrops / Muscle Fibers, Skeletal / Reptilian Proteins / Phospholipases A2 / Group II Phospholipases A2 / Phospholipase A2 Inhibitors / Indoles / Keto Acids / Acetates Limits: Animals Language: En Journal: Biochim Biophys Acta Gen Subj Year: 2021 Document type: Article Affiliation country: Brazil Country of publication: Netherlands

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Bothrops / Muscle Fibers, Skeletal / Reptilian Proteins / Phospholipases A2 / Group II Phospholipases A2 / Phospholipase A2 Inhibitors / Indoles / Keto Acids / Acetates Limits: Animals Language: En Journal: Biochim Biophys Acta Gen Subj Year: 2021 Document type: Article Affiliation country: Brazil Country of publication: Netherlands