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The Effect of Core Replacement on S64315, a Selective MCL-1 Inhibitor, and Its Analogues.
Sipos, Szabolcs; Bálint, Balázs; Szabó, Zoltán B; Ondi, Levente; Csékei, Márton; Szlávik, Zoltán; Proszenyák, Ágnes; Murray, James B; Davidson, James; Chen, Ijen; Dokurno, Pawel; Surgenor, Allan E; Pedder, Christopher; Hubbard, Roderick E; Maragno, Ana-Leticia; Chanrion, Maia; Colland, Frederic; Geneste, Olivier; Kotschy, András.
Affiliation
  • Sipos S; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
  • Bálint B; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
  • Szabó ZB; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
  • Ondi L; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
  • Csékei M; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
  • Szlávik Z; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
  • Proszenyák Á; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
  • Murray JB; Vernalis (R&D) Ltd., Granta Park, Cambridge CB21 6GB, UK.
  • Davidson J; Vernalis (R&D) Ltd., Granta Park, Cambridge CB21 6GB, UK.
  • Chen I; Vernalis (R&D) Ltd., Granta Park, Cambridge CB21 6GB, UK.
  • Dokurno P; Vernalis (R&D) Ltd., Granta Park, Cambridge CB21 6GB, UK.
  • Surgenor AE; Vernalis (R&D) Ltd., Granta Park, Cambridge CB21 6GB, UK.
  • Pedder C; Vernalis (R&D) Ltd., Granta Park, Cambridge CB21 6GB, UK.
  • Hubbard RE; Vernalis (R&D) Ltd., Granta Park, Cambridge CB21 6GB, UK.
  • Maragno AL; Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France.
  • Chanrion M; Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France.
  • Colland F; Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France.
  • Geneste O; Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France.
  • Kotschy A; Servier Research Institute of Medicinal Chemistry, Záhony u. 7., H-1031 Budapest, Hungary.
ACS Omega ; 6(34): 22073-22102, 2021 Aug 31.
Article in En | MEDLINE | ID: mdl-34497901

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Omega Year: 2021 Document type: Article Affiliation country: Hungary Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Omega Year: 2021 Document type: Article Affiliation country: Hungary Country of publication: United States