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Discovery and radiosensitization research of ursolic acid derivatives as SENP1 inhibitors.
Wei, Huiqiang; Guo, Jianghong; Sun, Xiao; Gou, Wenfeng; Ning, Hongxin; Fang, Zhennan; Liu, Qiang; Hou, Wenbin; Li, Yiliang.
Affiliation
  • Wei H; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China.
  • Guo J; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China.
  • Sun X; School of Traditional Chinese Medicine, Guangdong Pharmaceutical University, Guangzhou, 510006, China.
  • Gou W; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China.
  • Ning H; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China.
  • Fang Z; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China.
  • Liu Q; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China. Electronic address: liuqiang@irm-cams.ac.cn.
  • Hou W; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China. Electronic address: houwenbin@irm-cams.ac.cn.
  • Li Y; Tianjin Key Laboratory of Radiation Medicine and Molecular Nuclear Medicine, Institute of Radiation Medicine, Peking Union Medical College & Chinese Academy of Medical Sciences, Tianjin, 300192, China. Electronic address: liyiliang@irm-cams.ac.cn.
Eur J Med Chem ; 227: 113918, 2022 Jan 05.
Article in En | MEDLINE | ID: mdl-34688014

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Triterpenes / Cysteine Endopeptidases / Cysteine Proteinase Inhibitors / Drug Discovery / Antineoplastic Agents Limits: Humans Language: En Journal: Eur J Med Chem Year: 2022 Document type: Article Affiliation country: China Country of publication: France

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Triterpenes / Cysteine Endopeptidases / Cysteine Proteinase Inhibitors / Drug Discovery / Antineoplastic Agents Limits: Humans Language: En Journal: Eur J Med Chem Year: 2022 Document type: Article Affiliation country: China Country of publication: France