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Discovery of a High-Affinity Fluoromethyl Analog of [11C]5-Cyano-N-(4-(4-methylpiperazin-1-yl)-2-(piperidin-1-yl)phenyl)furan-2-carboxamide ([11C]CPPC) and Their Comparison in Mouse and Monkey as Colony-Stimulating Factor 1 Receptor Positron Emission Tomography Radioligands.
Altomonte, Stefano; Yan, Xuefeng; Morse, Cheryl L; Liow, Jeih-San; Jenkins, Madeline D; Montero Santamaria, Jose A; Zoghbi, Sami S; Innis, Robert B; Pike, Victor W.
Affiliation
  • Altomonte S; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Yan X; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Morse CL; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Liow JS; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Jenkins MD; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Montero Santamaria JA; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Zoghbi SS; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Innis RB; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
  • Pike VW; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health Building 10, B3 C346A, 10 Center Drive, Bethesda, Maryland 20892, United States.
ACS Pharmacol Transl Sci ; 6(4): 614-632, 2023 Apr 14.
Article in En | MEDLINE | ID: mdl-37082755

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Prognostic_studies Language: En Journal: ACS Pharmacol Transl Sci Year: 2023 Document type: Article Affiliation country: United States Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Prognostic_studies Language: En Journal: ACS Pharmacol Transl Sci Year: 2023 Document type: Article Affiliation country: United States Country of publication: United States