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From PERK to RIPK1: Design, synthesis and evaluation of novel potent and selective necroptosis inhibitors.
Scarpellini, Camilla; Valembois, Sophie; Goossens, Kenneth; Vadi, Mike; Lanthier, Caroline; Klejborowska, Greta; Van Der Veken, Pieter; De Winter, Hans; Bertrand, Mathieu J M; Augustyns, Koen.
Affiliation
  • Scarpellini C; Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Antwerp, Belgium.
  • Valembois S; Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Antwerp, Belgium.
  • Goossens K; Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Antwerp, Belgium.
  • Vadi M; Vlaams Instituut voor Biotechnologie (VIB) Center for Inflammation Research, Ghent, Belgium.
  • Lanthier C; Laboratory Cell Death and Inflammation, Department of Biomedical Molecular Biology, Ghent University, Ghent, Belgium.
  • Klejborowska G; Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Antwerp, Belgium.
  • Van Der Veken P; Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Antwerp, Belgium.
  • De Winter H; Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Antwerp, Belgium.
  • Bertrand MJM; Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Antwerp, Belgium.
  • Augustyns K; Vlaams Instituut voor Biotechnologie (VIB) Center for Inflammation Research, Ghent, Belgium.
Front Chem ; 11: 1160164, 2023.
Article in En | MEDLINE | ID: mdl-37090247

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: Front Chem Year: 2023 Document type: Article Affiliation country: Belgium Country of publication: Switzerland

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: Front Chem Year: 2023 Document type: Article Affiliation country: Belgium Country of publication: Switzerland