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3-Amido-3-aryl-piperidines: A Novel Class of Potent, Selective, and Orally Active GlyT1 Inhibitors.
Pinard, Emmanuel; Alberati, Daniela; Alvarez-Sanchez, Ruben; Brom, Virginie; Burner, Serge; Fischer, Holger; Hauser, Nicole; Kolczewski, Sabine; Lengyel, Judith; Mory, Roland; Saladin, Christian; Schulz-Gasch, Tanja; Stalder, Henri.
Afiliación
  • Pinard E; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Alberati D; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Alvarez-Sanchez R; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Brom V; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Burner S; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Fischer H; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Hauser N; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Kolczewski S; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Lengyel J; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Mory R; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Saladin C; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Schulz-Gasch T; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
  • Stalder H; Pharmaceutical Research Basel, F. Hoffmann-La Roche Ltd. , CH-4070 Basel, Switzerland.
ACS Med Chem Lett ; 5(4): 428-33, 2014 Apr 10.
Article en En | MEDLINE | ID: mdl-24900853

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2014 Tipo del documento: Article País de afiliación: Suiza Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2014 Tipo del documento: Article País de afiliación: Suiza Pais de publicación: Estados Unidos