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Identification and characterization of a selective allosteric antagonist of human P2X4 receptor channels.
Ase, Ariel R; Honson, Nicolette S; Zaghdane, Helmi; Pfeifer, Tom A; Séguéla, Philippe.
Afiliación
  • Ase AR; Montreal Neurological Institute, Alan Edwards Centre for Research on Pain, Department of Neurology and Neurosurgery, McGill University, Montreal, Canada (A.R.A., P.S.); Screening Division, The Centre for Drug Research and Discovery, Vancouver, Canada (N.S.H., T.A.P.); and Zamboni Chemical Solutions,
  • Honson NS; Montreal Neurological Institute, Alan Edwards Centre for Research on Pain, Department of Neurology and Neurosurgery, McGill University, Montreal, Canada (A.R.A., P.S.); Screening Division, The Centre for Drug Research and Discovery, Vancouver, Canada (N.S.H., T.A.P.); and Zamboni Chemical Solutions,
  • Zaghdane H; Montreal Neurological Institute, Alan Edwards Centre for Research on Pain, Department of Neurology and Neurosurgery, McGill University, Montreal, Canada (A.R.A., P.S.); Screening Division, The Centre for Drug Research and Discovery, Vancouver, Canada (N.S.H., T.A.P.); and Zamboni Chemical Solutions,
  • Pfeifer TA; Montreal Neurological Institute, Alan Edwards Centre for Research on Pain, Department of Neurology and Neurosurgery, McGill University, Montreal, Canada (A.R.A., P.S.); Screening Division, The Centre for Drug Research and Discovery, Vancouver, Canada (N.S.H., T.A.P.); and Zamboni Chemical Solutions,
  • Séguéla P; Montreal Neurological Institute, Alan Edwards Centre for Research on Pain, Department of Neurology and Neurosurgery, McGill University, Montreal, Canada (A.R.A., P.S.); Screening Division, The Centre for Drug Research and Discovery, Vancouver, Canada (N.S.H., T.A.P.); and Zamboni Chemical Solutions,
Mol Pharmacol ; 87(4): 606-16, 2015 Apr.
Article en En | MEDLINE | ID: mdl-25597706

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Compuestos de Fenilurea / Receptores Purinérgicos P2X4 / Antagonistas del Receptor Purinérgico P2X / Aminopiridinas Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Animals / Humans Idioma: En Revista: Mol Pharmacol Año: 2015 Tipo del documento: Article Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Compuestos de Fenilurea / Receptores Purinérgicos P2X4 / Antagonistas del Receptor Purinérgico P2X / Aminopiridinas Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Animals / Humans Idioma: En Revista: Mol Pharmacol Año: 2015 Tipo del documento: Article Pais de publicación: Estados Unidos