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EPI-001 is a selective peroxisome proliferator-activated receptor-gamma modulator with inhibitory effects on androgen receptor expression and activity in prostate cancer.
Brand, Lucas J; Olson, Margaret E; Ravindranathan, Preethi; Guo, Hong; Kempema, Aaron M; Andrews, Timothy E; Chen, Xiaoli; Raj, Ganesh V; Harki, Daniel A; Dehm, Scott M.
Afiliación
  • Brand LJ; Graduate Program in Microbiology, Immunology, and Cancer Biology, University of Minnesota, Minneapolis, MN, USA.
  • Olson ME; Masonic Cancer Center, University of Minnesota, Minneapolis, MN, USA.
  • Ravindranathan P; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, MN, USA.
  • Guo H; Department of Urology, University of Texas Southwestern Medical Center, Dallas, Texas, USA.
  • Kempema AM; Department of Food Science and Nutrition, University of Minnesota, Minneapolis, MN, USA.
  • Andrews TE; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, MN, USA.
  • Chen X; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, MN, USA.
  • Raj GV; Department of Food Science and Nutrition, University of Minnesota, Minneapolis, MN, USA.
  • Harki DA; Department of Urology, University of Texas Southwestern Medical Center, Dallas, Texas, USA.
  • Dehm SM; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, MN, USA.
Oncotarget ; 6(6): 3811-24, 2015 Feb 28.
Article en En | MEDLINE | ID: mdl-25669987

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Compuestos de Bencidrilo / Receptores Androgénicos / Clorhidrinas / Antagonistas de Receptores Androgénicos Límite: Humans / Male Idioma: En Revista: Oncotarget Año: 2015 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Compuestos de Bencidrilo / Receptores Androgénicos / Clorhidrinas / Antagonistas de Receptores Androgénicos Límite: Humans / Male Idioma: En Revista: Oncotarget Año: 2015 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos