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Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3.
Li, Lei; Shao, Xia; Cole, Erin L; Ohnmacht, Stephan A; Ferrari, Valentina; Hong, Young T; Williamson, David J; Fryer, Tim D; Quesada, Carole A; Sherman, Phillip; Riss, Patrick J; Scott, Peter J H; Aigbirhio, Franklin I.
Afiliación
  • Li L; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
  • Shao X; Division of Nuclear Medicine, Department of Radiology, The University of Michigan Medical School , Ann Arbor, Michigan 48109, United States.
  • Cole EL; Division of Nuclear Medicine, Department of Radiology, The University of Michigan Medical School , Ann Arbor, Michigan 48109, United States.
  • Ohnmacht SA; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
  • Ferrari V; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
  • Hong YT; Laboratory for Molecular Imaging, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
  • Williamson DJ; Laboratory for Molecular Imaging, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
  • Fryer TD; Laboratory for Molecular Imaging, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
  • Quesada CA; Division of Nuclear Medicine, Department of Radiology, The University of Michigan Medical School , Ann Arbor, Michigan 48109, United States.
  • Sherman P; Division of Nuclear Medicine, Department of Radiology, The University of Michigan Medical School , Ann Arbor, Michigan 48109, United States.
  • Riss PJ; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
  • Scott PJ; Division of Nuclear Medicine, Department of Radiology, The University of Michigan Medical School , Ann Arbor, Michigan 48109, United States ; The Interdepartmental Program in Medicinal Chemistry, The University of Michigan , Ann Arbor, Michigan 48109, United States.
  • Aigbirhio FI; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K. ; Laboratory for Molecular Imaging, Wolfson Brain Imaging Centre, University of Cambridge , Cambridge CB2 1TN, U.K.
ACS Med Chem Lett ; 6(5): 548-52, 2015 May 14.
Article en En | MEDLINE | ID: mdl-26005531

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2015 Tipo del documento: Article País de afiliación: Reino Unido Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2015 Tipo del documento: Article País de afiliación: Reino Unido Pais de publicación: Estados Unidos