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Multiple spatially related pharmacophores define small molecule inhibitors of OLIG2 in glioblastoma.
Tsigelny, Igor F; Mukthavaram, Rajesh; Kouznetsova, Valentina L; Chao, Ying; Babic, Ivan; Nurmemmedov, Elmar; Pastorino, Sandra; Jiang, Pengfei; Calligaris, David; Agar, Nathalie; Scadeng, Miriam; Pingle, Sandeep C; Wrasidlo, Wolfgang; Makale, Milan T; Kesari, Santosh.
Afiliación
  • Tsigelny IF; Department of Neurosciences, University of California San Diego, La Jolla, CA, USA.
  • Mukthavaram R; San Diego Supercomputer Center, University of California San Diego, La Jolla, CA, USA.
  • Kouznetsova VL; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
  • Chao Y; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
  • Babic I; San Diego Supercomputer Center, University of California San Diego, La Jolla, CA, USA.
  • Nurmemmedov E; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
  • Pastorino S; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
  • Jiang P; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
  • Calligaris D; The Scripps Research Institute, La Jolla, CA, USA.
  • Agar N; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
  • Scadeng M; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
  • Pingle SC; Harvard Medical School, Department of Neurosurgery, Brigham and Women's Hospital, Boston, MA, USA.
  • Wrasidlo W; Harvard Medical School, Department of Neurosurgery, Brigham and Women's Hospital, Boston, MA, USA.
  • Makale MT; FMRI Research Center, Department of Radiology, University of California San Diego, La Jolla, CA, USA.
  • Kesari S; Translational Neuro-oncology Laboratories, Moores Cancer Center, University of California San Diego, La Jolla, CA, USA.
Oncotarget ; 8(14): 22370-22384, 2017 Apr 04.
Article en En | MEDLINE | ID: mdl-26517684

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias Encefálicas / Diseño de Fármacos / Glioblastoma / Factores de Transcripción con Motivo Hélice-Asa-Hélice Básico / Terapia Molecular Dirigida / Guanidinas / Proteínas del Tejido Nervioso / Antineoplásicos Tipo de estudio: Prognostic_studies Límite: Animals / Humans Idioma: En Revista: Oncotarget Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias Encefálicas / Diseño de Fármacos / Glioblastoma / Factores de Transcripción con Motivo Hélice-Asa-Hélice Básico / Terapia Molecular Dirigida / Guanidinas / Proteínas del Tejido Nervioso / Antineoplásicos Tipo de estudio: Prognostic_studies Límite: Animals / Humans Idioma: En Revista: Oncotarget Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos