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Diclofenac and Its Acyl Glucuronide: Determination of In Vivo Exposure in Human Subjects and Characterization as Human Drug Transporter Substrates In Vitro.
Zhang, Yueping; Han, Yong-Hae; Putluru, Siva Prasad; Matta, Murali Krishna; Kole, Prashant; Mandlekar, Sandhya; Furlong, Michael T; Liu, Tongtong; Iyer, Ramaswamy A; Marathe, Punit; Yang, Zheng; Lai, Yurong; Rodrigues, A David.
Afiliación
  • Zhang Y; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Han YH; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Putluru SP; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Matta MK; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Kole P; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Mandlekar S; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Furlong MT; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Liu T; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Iyer RA; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Marathe P; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Yang Z; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
  • Lai Y; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey yurong.lai@bms.com.
  • Rodrigues AD; Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Princeton, New Jersey.
Drug Metab Dispos ; 44(3): 320-8, 2016 Mar.
Article en En | MEDLINE | ID: mdl-26714763

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Transporte Biológico / Diclofenaco / Glucurónidos / Transportadores de Anión Orgánico Límite: Adult / Humans / Male Idioma: En Revista: Drug Metab Dispos Asunto de la revista: FARMACOLOGIA Año: 2016 Tipo del documento: Article Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Transporte Biológico / Diclofenaco / Glucurónidos / Transportadores de Anión Orgánico Límite: Adult / Humans / Male Idioma: En Revista: Drug Metab Dispos Asunto de la revista: FARMACOLOGIA Año: 2016 Tipo del documento: Article Pais de publicación: Estados Unidos