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The use of isomeric testosterone dimers to explore allosteric effects in substrate binding to cytochrome P450 CYP3A4.
Denisov, Ilia G; Mak, Piotr J; Grinkova, Yelena V; Bastien, Dominic; Bérubé, Gervais; Sligar, Stephen G; Kincaid, James R.
Afiliación
  • Denisov IG; Department of Biochemistry, University of Illinois, Urbana, IL 61801, United States. Electronic address: denisov@illinois.edu.
  • Mak PJ; Department of Chemistry, Marquette University, Milwaukee, WI 53233, United States. Electronic address: piotr.mak@marquette.edu.
  • Grinkova YV; Department of Biochemistry, University of Illinois, Urbana, IL 61801, United States. Electronic address: grinkova@illinois.edu.
  • Bastien D; Département de chimie, biochimie et physique, Université du Québec à Trois-Rivières, Trois-Rivières, Québec G9A 5H7, Canada. Electronic address: Dominic.Bastien@uqtr.ca.
  • Bérubé G; Département de chimie, biochimie et physique, Université du Québec à Trois-Rivières, Trois-Rivières, Québec G9A 5H7, Canada. Electronic address: Gervais.Berube@uqtr.ca.
  • Sligar SG; Department of Biochemistry, University of Illinois, Urbana, IL 61801, United States; Department of Chemistry, University of Illinois, Urbana, IL 61801, United States. Electronic address: s-sligar@illinois.edu.
  • Kincaid JR; Department of Chemistry, Marquette University, Milwaukee, WI 53233, United States. Electronic address: james.kincaid@marquette.edu.
J Inorg Biochem ; 158: 77-85, 2016 05.
Article en En | MEDLINE | ID: mdl-26774838

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Testosterona / Citocromo P-450 CYP3A Límite: Humans Idioma: En Revista: J Inorg Biochem Año: 2016 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Testosterona / Citocromo P-450 CYP3A Límite: Humans Idioma: En Revista: J Inorg Biochem Año: 2016 Tipo del documento: Article