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Design and Structural Characterization of Potent and Selective Inhibitors of Phosphatidylinositol 4 Kinase IIIß.
Rutaganira, Florentine U; Fowler, Melissa L; McPhail, Jacob A; Gelman, Michael A; Nguyen, Khanh; Xiong, Anming; Dornan, Gillian L; Tavshanjian, Brandon; Glenn, Jeffrey S; Shokat, Kevan M; Burke, John E.
Afiliación
  • Rutaganira FU; Howard Hughes Medical Institute and Department of Cellular and Molecular Pharmacology, University of California, San Francisco (UCSF) , San Francisco, California 94143, United States.
  • Fowler ML; Department of Biochemistry and Microbiology, University of Victoria , Victoria, BC V8W 2Y2, Canada.
  • McPhail JA; Department of Biochemistry and Microbiology, University of Victoria , Victoria, BC V8W 2Y2, Canada.
  • Gelman MA; Department of Medicine and Department of Microbiology & Immunology, Stanford University , Palo Alto, California 94305, United States.
  • Nguyen K; Department of Medicine and Department of Microbiology & Immunology, Stanford University , Palo Alto, California 94305, United States.
  • Xiong A; Department of Medicine and Department of Microbiology & Immunology, Stanford University , Palo Alto, California 94305, United States.
  • Dornan GL; Department of Biochemistry and Microbiology, University of Victoria , Victoria, BC V8W 2Y2, Canada.
  • Tavshanjian B; Howard Hughes Medical Institute and Department of Cellular and Molecular Pharmacology, University of California, San Francisco (UCSF) , San Francisco, California 94143, United States.
  • Glenn JS; Department of Medicine and Department of Microbiology & Immunology, Stanford University , Palo Alto, California 94305, United States.
  • Shokat KM; Veterans Administration Medical Center , Palo Alto, California 94304, United States.
  • Burke JE; Howard Hughes Medical Institute and Department of Cellular and Molecular Pharmacology, University of California, San Francisco (UCSF) , San Francisco, California 94143, United States.
J Med Chem ; 59(5): 1830-9, 2016 Mar 10.
Article en En | MEDLINE | ID: mdl-26885694

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Antivirales / Diseño de Fármacos / Fosfotransferasas (Aceptor de Grupo Alcohol) / Inhibidores de Proteínas Quinasas Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Antivirales / Diseño de Fármacos / Fosfotransferasas (Aceptor de Grupo Alcohol) / Inhibidores de Proteínas Quinasas Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos