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Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer.
Bassetto, Marcella; Ferla, Salvatore; Pertusati, Fabrizio; Kandil, Sahar; Westwell, Andrew D; Brancale, Andrea; McGuigan, Christopher.
Afiliación
  • Bassetto M; School of Pharmacy and Pharmaceutical Sciences, Redwood Building, King Edward VII Avenue, CF10 3NB, Cardiff, Wales, UK.
  • Ferla S; School of Pharmacy and Pharmaceutical Sciences, Redwood Building, King Edward VII Avenue, CF10 3NB, Cardiff, Wales, UK. Electronic address: Ferlas1@cardiff.ac.uk.
  • Pertusati F; School of Pharmacy and Pharmaceutical Sciences, Redwood Building, King Edward VII Avenue, CF10 3NB, Cardiff, Wales, UK.
  • Kandil S; School of Pharmacy and Pharmaceutical Sciences, Redwood Building, King Edward VII Avenue, CF10 3NB, Cardiff, Wales, UK.
  • Westwell AD; School of Pharmacy and Pharmaceutical Sciences, Redwood Building, King Edward VII Avenue, CF10 3NB, Cardiff, Wales, UK.
  • Brancale A; School of Pharmacy and Pharmaceutical Sciences, Redwood Building, King Edward VII Avenue, CF10 3NB, Cardiff, Wales, UK.
  • McGuigan C; School of Pharmacy and Pharmaceutical Sciences, Redwood Building, King Edward VII Avenue, CF10 3NB, Cardiff, Wales, UK.
Eur J Med Chem ; 118: 230-43, 2016 Aug 08.
Article en En | MEDLINE | ID: mdl-27131065

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Feniltiohidantoína / Neoplasias de la Próstata / Compuestos de Tosilo / Diseño de Fármacos / Anilidas / Nitrilos Límite: Humans / Male Idioma: En Revista: Eur J Med Chem Año: 2016 Tipo del documento: Article País de afiliación: Reino Unido Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Feniltiohidantoína / Neoplasias de la Próstata / Compuestos de Tosilo / Diseño de Fármacos / Anilidas / Nitrilos Límite: Humans / Male Idioma: En Revista: Eur J Med Chem Año: 2016 Tipo del documento: Article País de afiliación: Reino Unido Pais de publicación: Francia