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Brain penetrant small molecule (18)F-GnRH receptor (GnRH-R) antagonists: Synthesis and preliminary positron emission tomography imaging in rats.
Olberg, Dag E; Bauer, Nadine; Andressen, Kjetil W; Hjørnevik, Trine; Cumming, Paul; Levy, Finn O; Klaveness, Jo; Haraldsen, Ira; Sutcliffe, Julie L.
Afiliación
  • Olberg DE; Norsk medisinsk syklotronsenter AS, Postboks 4950 Nydalen, 0424 Oslo, Norway; School of Pharmacy, University of Oslo, P.O.Box 1068, Blindern, 0316 Oslo, Norway. Electronic address: dag.erlend.olberg@petsenteret.no.
  • Bauer N; Department of Biomedical Engineering, University of California Davis, Davis, CA, USA.
  • Andressen KW; Department of Pharmacology, Faculty of Medicine, University of Oslo and Oslo, University Hospital, Oslo, Norway; K.G. Jebsen Cardiac Research Centre and Center for Heart Failure Research, Faculty of Medicine, University of Oslo, Oslo, Norway.
  • Hjørnevik T; The Intervention Centre, Oslo University Hospital, PO 4950, Nydalen, 0424 Oslo, Norway.
  • Cumming P; Department of Neuropsychiatry and Psychosomatic Medicine, Oslo University Hospital, Oslo, Norway; School of Psychology and Conselling, Queensland University of Technology and QIMR Berghofer, Brisbane, Australia.
  • Levy FO; Department of Pharmacology, Faculty of Medicine, University of Oslo and Oslo, University Hospital, Oslo, Norway; K.G. Jebsen Cardiac Research Centre and Center for Heart Failure Research, Faculty of Medicine, University of Oslo, Oslo, Norway.
  • Klaveness J; School of Pharmacy, University of Oslo, P.O.Box 1068, Blindern, 0316 Oslo, Norway.
  • Haraldsen I; Department of Neuropsychiatry and Psychosomatic Medicine, Oslo University Hospital, Oslo, Norway.
  • Sutcliffe JL; Department of Biomedical Engineering, University of California Davis, Davis, CA, USA; Division of Hematology/Oncology, Department of Internal Medicine, University of California Davis, Sacramento, CA; Center for Molecular and Genomic Imaging, University of California Davis, Davis, CA; Radiochemistry
Nucl Med Biol ; 43(8): 478-89, 2016 08.
Article en En | MEDLINE | ID: mdl-27236283

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Encéfalo / Radioisótopos de Flúor / Receptores LHRH / Furanos Límite: Animals Idioma: En Revista: Nucl Med Biol Asunto de la revista: BIOLOGIA / MEDICINA NUCLEAR Año: 2016 Tipo del documento: Article Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Encéfalo / Radioisótopos de Flúor / Receptores LHRH / Furanos Límite: Animals Idioma: En Revista: Nucl Med Biol Asunto de la revista: BIOLOGIA / MEDICINA NUCLEAR Año: 2016 Tipo del documento: Article Pais de publicación: Estados Unidos