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1-(4-[18F]Fluorobenzyl)-4-[(tetrahydrofuran-2-yl)methyl]piperazine: A Novel Suitable Radioligand with Low Lipophilicity for Imaging σ1 Receptors in the Brain.
He, Yingfang; Xie, Fang; Ye, Jiajun; Deuther-Conrad, Winnie; Cui, Bixiao; Wang, Liang; Lu, Jie; Steinbach, Jörg; Brust, Peter; Huang, Yiyun; Lu, Jie; Jia, Hongmei.
Afiliación
  • He Y; Key Laboratory of Radiopharmaceuticals (Beijing Normal University), Ministry of Education, College of Chemistry, Beijing Normal University , Beijing, China.
  • Xie F; Key Laboratory of Radiopharmaceuticals (Beijing Normal University), Ministry of Education, College of Chemistry, Beijing Normal University , Beijing, China.
  • Ye J; Key Laboratory of Radiopharmaceuticals (Beijing Normal University), Ministry of Education, College of Chemistry, Beijing Normal University , Beijing, China.
  • Deuther-Conrad W; Helmholtz-Zentrum Dresden-Rossendorf , Institute of Radiopharmaceutical Cancer Research, Department of Neuroradiopharmaceuticals, 04318 Leipzig, Germany.
  • Cui B; Department of Nuclear Medicine, Xuanwu Hospital Capital Medical University , Beijing, China.
  • Wang L; Key Laboratory of Radiopharmaceuticals (Beijing Normal University), Ministry of Education, College of Chemistry, Beijing Normal University , Beijing, China.
  • Lu J; Key Laboratory of Radiopharmaceuticals (Beijing Normal University), Ministry of Education, College of Chemistry, Beijing Normal University , Beijing, China.
  • Steinbach J; Helmholtz-Zentrum Dresden-Rossendorf , Institute of Radiopharmaceutical Cancer Research, Department of Neuroradiopharmaceuticals, 04318 Leipzig, Germany.
  • Brust P; Helmholtz-Zentrum Dresden-Rossendorf , Institute of Radiopharmaceutical Cancer Research, Department of Neuroradiopharmaceuticals, 04318 Leipzig, Germany.
  • Huang Y; Yale PET Center, Department of Radiology and Biomedical Imaging, Yale University School of Medicine , New Haven, Connecticut 06520-8048, United States.
  • Lu J; Department of Nuclear Medicine, Xuanwu Hospital Capital Medical University , Beijing, China.
  • Jia H; Key Laboratory of Radiopharmaceuticals (Beijing Normal University), Ministry of Education, College of Chemistry, Beijing Normal University , Beijing, China.
J Med Chem ; 60(10): 4161-4172, 2017 05 25.
Article en En | MEDLINE | ID: mdl-28409931

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperazinas / Encéfalo / Radioisótopos de Flúor / Receptores sigma Límite: Animals Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: China Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperazinas / Encéfalo / Radioisótopos de Flúor / Receptores sigma Límite: Animals Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: China Pais de publicación: Estados Unidos