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Substituted N-Phenyl-5-(2-(phenylamino)thiazol-4-yl)isoxazole-3-carboxamides Are Valuable Antitubercular Candidates that Evade Innate Efflux Machinery.
Azzali, Elisa; Machado, Diana; Kaushik, Amit; Vacondio, Federica; Flisi, Sara; Cabassi, Clotilde Silvia; Lamichhane, Gyanu; Viveiros, Miguel; Costantino, Gabriele; Pieroni, Marco.
Afiliación
  • Azzali E; Centro Interdipartimentale Misure (CIM) 'G. Casnati', University of Parma , Parco Area delle Scienze 23/A, 43124 Parma, Italy.
  • Machado D; Global Health and Tropical Medicine, GHTM, Instituto de Higiene e Medicina Tropical, IHMT, Universidade Nova de Lisboa, UNL , Rua da Junqueira, 100, 1349-008 Lisbon, Portugal.
  • Kaushik A; Center for Tuberculosis Research, Department of Medicine, Johns Hopkins University , 1503 East Jefferson Street, Baltimore, Maryland 21231-1002, United States.
  • Vacondio F; Taskforce to Study Resistance Emergence & Antimicrobial development Technology, Department of Medicine, Johns Hopkins University , Baltimore, Maryland 21287, United States.
  • Cabassi CS; Department of Veterinary Science, University of Parma , via del Taglio 10, 43126 Parma, Italy.
  • Lamichhane G; Department of Veterinary Science, University of Parma , via del Taglio 10, 43126 Parma, Italy.
  • Viveiros M; Center for Tuberculosis Research, Department of Medicine, Johns Hopkins University , 1503 East Jefferson Street, Baltimore, Maryland 21231-1002, United States.
  • Costantino G; Taskforce to Study Resistance Emergence & Antimicrobial development Technology, Department of Medicine, Johns Hopkins University , Baltimore, Maryland 21287, United States.
  • Pieroni M; Global Health and Tropical Medicine, GHTM, Instituto de Higiene e Medicina Tropical, IHMT, Universidade Nova de Lisboa, UNL , Rua da Junqueira, 100, 1349-008 Lisbon, Portugal.
J Med Chem ; 60(16): 7108-7122, 2017 08 24.
Article en En | MEDLINE | ID: mdl-28749666

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tiazoles / Isoxazoles / Antituberculosos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tiazoles / Isoxazoles / Antituberculosos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia Pais de publicación: Estados Unidos