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Novel xanthone-polyamine conjugates as catalytic inhibitors of human topoisomerase IIα.
Minniti, Elirosa; Byl, Jo Ann W; Riccardi, Laura; Sissi, Claudia; Rosini, Michela; De Vivo, Marco; Minarini, Anna; Osheroff, Neil.
Afiliación
  • Minniti E; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, Via Belmeloro 6, 40126 Bologna, Italy; Laboratory of Molecular Modeling and Drug Discovery, Istituto Italiano di Tecnologia, Via Morego 30, 16163 Genova, Italy.
  • Byl JAW; Department of Biochemistry, Vanderbilt University School of Medicine, Nashville, TN 37232-0146, USA.
  • Riccardi L; Laboratory of Molecular Modeling and Drug Discovery, Istituto Italiano di Tecnologia, Via Morego 30, 16163 Genova, Italy.
  • Sissi C; Department of Pharmaceutical and Pharmacological Sciences, University of Padova, Via Marzolo 5, 35131 Padova, Italy.
  • Rosini M; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, Via Belmeloro 6, 40126 Bologna, Italy.
  • De Vivo M; Laboratory of Molecular Modeling and Drug Discovery, Istituto Italiano di Tecnologia, Via Morego 30, 16163 Genova, Italy; IAS-5/INM-9 Computational Biomedicine, Forschungszentrum Jülich, Wilhelm-Johnen-Straße, 52428 Jülich, Germany.
  • Minarini A; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, Via Belmeloro 6, 40126 Bologna, Italy. Electronic address: anna.minarini@unibo.it.
  • Osheroff N; Department of Biochemistry, Vanderbilt University School of Medicine, Nashville, TN 37232-0146, USA; Department of Medicine (Hematology/Oncology), Vanderbilt University School of Medicine, Nashville, TN 37232-6307, USA; VA Tennessee Valley Healthcare System, Nashville, TN 37212, USA. Electronic addr
Bioorg Med Chem Lett ; 27(20): 4687-4693, 2017 10 15.
Article en En | MEDLINE | ID: mdl-28919339

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Poliaminas / Xantonas / Proteínas de Unión al ADN / Inhibidores de Topoisomerasa II Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Poliaminas / Xantonas / Proteínas de Unión al ADN / Inhibidores de Topoisomerasa II Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia