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[Carboxyl-11 C]Labelling of Four High-Affinity cPLA2α Inhibitors and Their Evaluation as Radioligands in Mice by Positron Emission Tomography.
Fisher, Martin J; McMurray, Lindsay; Lu, Shuiyu; Morse, Cheryl L; Liow, Jeih-San; Zoghbi, Sami S; Kowalski, Aneta; Tye, George L; Innis, Robert B; Aigbirhio, Franklin I; Pike, Victor W.
Afiliación
  • Fisher MJ; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge, Cambridge Biomedical Campus, Cambridge, CB2 0QQ, UK.
  • McMurray L; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge, Cambridge Biomedical Campus, Cambridge, CB2 0QQ, UK.
  • Lu S; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
  • Morse CL; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
  • Liow JS; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
  • Zoghbi SS; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
  • Kowalski A; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
  • Tye GL; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
  • Innis RB; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
  • Aigbirhio FI; Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre, University of Cambridge, Cambridge Biomedical Campus, Cambridge, CB2 0QQ, UK.
  • Pike VW; Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, 10 Center Drive, Room B3C346, Bethesda, MD 20892, USA.
ChemMedChem ; 13(2): 138-146, 2018 01 22.
Article en En | MEDLINE | ID: mdl-29232493

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Radiofármacos / Inhibidores Enzimáticos / Fosfolipasas A2 Grupo IV Límite: Animals / Humans Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Reino Unido Pais de publicación: Alemania

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Radiofármacos / Inhibidores Enzimáticos / Fosfolipasas A2 Grupo IV Límite: Animals / Humans Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Reino Unido Pais de publicación: Alemania