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Small Molecule Inhibitor that Stabilizes the Autoinhibited Conformation of the Oncogenic Tyrosine Phosphatase SHP2.
Wu, Xiaoqin; Xu, Gang; Li, Xiaobo; Xu, Weiren; Li, Qianjin; Liu, Wei; Kirby, Karen A; Loh, Mignon L; Li, Jun; Sarafianos, Stefan G; Qu, Cheng-Kui.
Afiliación
  • Wu X; Department of Pediatrics, Division of Hematology/Oncology, Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta , Emory University School of Medicine , Atlanta , Georgia 30322 , United States.
  • Xu G; Department of Medicine, Division of Hematology and Oncology, Case Comprehensive Cancer Center , Case Western Reserve University , Cleveland , Ohio 44106 , United States.
  • Li X; Department of Pediatrics, Division of Hematology/Oncology, Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta , Emory University School of Medicine , Atlanta , Georgia 30322 , United States.
  • Xu W; Department of Medicine, Division of Hematology and Oncology, Case Comprehensive Cancer Center , Case Western Reserve University , Cleveland , Ohio 44106 , United States.
  • Li Q; Department of Medicine, Division of Hematology and Oncology, Case Comprehensive Cancer Center , Case Western Reserve University , Cleveland , Ohio 44106 , United States.
  • Liu W; Department of Pediatrics, Division of Hematology/Oncology, Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta , Emory University School of Medicine , Atlanta , Georgia 30322 , United States.
  • Kirby KA; Department of Medicine, Division of Hematology and Oncology, Case Comprehensive Cancer Center , Case Western Reserve University , Cleveland , Ohio 44106 , United States.
  • Loh ML; Department of Pediatrics, Laboratory of Biochemical Pharmacology , Emory University School of Medicine , Atlanta , Georgia 30322 , United States.
  • Li J; Department of Pediatrics, Division of Pediatric Hematology-Oncology , University of California, San Francisco , San Francisco , California 94122 , United States.
  • Sarafianos SG; School of Pharmacy , Anhui Medical University , Hefei 230032 , China.
  • Qu CK; Department of Pediatrics, Laboratory of Biochemical Pharmacology , Emory University School of Medicine , Atlanta , Georgia 30322 , United States.
J Med Chem ; 62(3): 1125-1137, 2019 02 14.
Article en En | MEDLINE | ID: mdl-30457860

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Proteína Tirosina Fosfatasa no Receptora Tipo 11 / Bibliotecas de Moléculas Pequeñas Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Proteína Tirosina Fosfatasa no Receptora Tipo 11 / Bibliotecas de Moléculas Pequeñas Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos