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Novel Aryloxyethyl Derivatives of 1-(1-Benzoylpiperidin-4-yl)methanamine as the Extracellular Regulated Kinases 1/2 (ERK1/2) Phosphorylation-Preferring Serotonin 5-HT1A Receptor-Biased Agonists with Robust Antidepressant-like Activity.
Sniecikowska, Joanna; Gluch-Lutwin, Monika; Bucki, Adam; Wieckowska, Anna; Siwek, Agata; Jastrzebska-Wiesek, Magdalena; Partyka, Anna; Wilczynska, Daria; Pytka, Karolina; Pociecha, Krzysztof; Cios, Agnieszka; Wyska, Elzbieta; Wesolowska, Anna; Pawlowski, Maciej; Varney, Mark A; Newman-Tancredi, Adrian; Kolaczkowski, Marcin.
Afiliación
  • Sniecikowska J; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Gluch-Lutwin M; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Bucki A; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Wieckowska A; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Siwek A; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Jastrzebska-Wiesek M; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Partyka A; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Wilczynska D; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Pytka K; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Pociecha K; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Cios A; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Wyska E; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Wesolowska A; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Pawlowski M; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
  • Varney MA; Neurolixis Inc. , 34145 Pacific Coast Highway #504 , Dana Point , 92629 California , United States.
  • Newman-Tancredi A; Neurolixis Inc. , 34145 Pacific Coast Highway #504 , Dana Point , 92629 California , United States.
  • Kolaczkowski M; Faculty of Pharmacy , Jagiellonian University Medical College , 9 Medyczna Street , 30-688 Kraków , Poland.
J Med Chem ; 62(5): 2750-2771, 2019 03 14.
Article en En | MEDLINE | ID: mdl-30721053

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperidinas / Agonistas de Receptores de Serotonina / Antidepresivos de Segunda Generación / Sistema de Señalización de MAP Quinasas / Receptor de Serotonina 5-HT1A Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Polonia Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperidinas / Agonistas de Receptores de Serotonina / Antidepresivos de Segunda Generación / Sistema de Señalización de MAP Quinasas / Receptor de Serotonina 5-HT1A Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Polonia Pais de publicación: Estados Unidos