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Agonist-selective NOP receptor phosphorylation correlates in vitro and in vivo and reveals differential post-activation signaling by chemically diverse agonists.
Mann, Anika; Moulédous, Lionel; Froment, Carine; O'Neill, Patrick R; Dasgupta, Pooja; Günther, Thomas; Brunori, Gloria; Kieffer, Brigitte L; Toll, Lawrence; Bruchas, Michael R; Zaveri, Nurulain T; Schulz, Stefan.
Afiliación
  • Mann A; Institute of Pharmacology and Toxicology, Jena University Hospital, Friedrich Schiller University Jena, Drackendorfer Str. 1, Jena 07747, Germany. anika.mann@med.uni-jena.de stefan.schulz@med.uni-jena.de.
  • Moulédous L; Research Center on Animal Cognition, Center for Integrative Biology, Toulouse University, CNRS, UPS, 31062 Toulouse Cedex 09, France.
  • Froment C; Institut de Pharmacologie et de Biologie Structurale, Université de Toulouse, CNRS, UPS, 31077 Toulouse Cedex 04, France.
  • O'Neill PR; Department of Anesthesiology, Washington University School of Medicine, St. Louis, MO 63110, USA.
  • Dasgupta P; Institute of Pharmacology and Toxicology, Jena University Hospital, Friedrich Schiller University Jena, Drackendorfer Str. 1, Jena 07747, Germany.
  • Günther T; Institute of Pharmacology and Toxicology, Jena University Hospital, Friedrich Schiller University Jena, Drackendorfer Str. 1, Jena 07747, Germany.
  • Brunori G; Biomedical Science Department, Charles E. Schmidt College of Medicine, Florida Atlantic University, Boca Raton, FL 33431, USA.
  • Kieffer BL; Douglas Research Center, Department of Psychiatry, Faculty of Medicine, McGill University, Montreal, QC H3A 1A1, Canada.
  • Toll L; Biomedical Science Department, Charles E. Schmidt College of Medicine, Florida Atlantic University, Boca Raton, FL 33431, USA.
  • Bruchas MR; Center for the Neurobiology of Addiction, Pain, and Emotion, Departments of Anesthesiology and Pharmacology, University of Washington, Seattle, WA 98195, USA.
  • Zaveri NT; Astraea Therapeutics LLC, Mountain View, CA 94043, USA.
  • Schulz S; Institute of Pharmacology and Toxicology, Jena University Hospital, Friedrich Schiller University Jena, Drackendorfer Str. 1, Jena 07747, Germany. anika.mann@med.uni-jena.de stefan.schulz@med.uni-jena.de.
Sci Signal ; 12(574)2019 03 26.
Article en En | MEDLINE | ID: mdl-30914485

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptores Opioides Límite: Animals / Humans Idioma: En Revista: Sci Signal Asunto de la revista: CIENCIA / FISIOLOGIA Año: 2019 Tipo del documento: Article Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptores Opioides Límite: Animals / Humans Idioma: En Revista: Sci Signal Asunto de la revista: CIENCIA / FISIOLOGIA Año: 2019 Tipo del documento: Article Pais de publicación: Estados Unidos