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Design, synthesis and biological evaluation of AT1 receptor blockers derived from 6-substituted aminocarbonyl benzimidazoles.
Wu, Zhuo; Anh, Nguyen Thi Phuong; Yan, Yi-Jia; Xia, Ming-Bao; Wang, Yan-Hui; Qiu, Yan; Chen, Zhi-Long.
Afiliación
  • Wu Z; Department of Pharmaceutical Science and Technology, College of Chemistry and Biology, Donghua University, Shanghai, 201620, China.
  • Anh NTP; Department of Pharmaceutical Science and Technology, College of Chemistry and Biology, Donghua University, Shanghai, 201620, China.
  • Yan YJ; Ningbo Dongmi Pharmaceutical Co., Ltd, Ningbo, 315899, China.
  • Xia MB; Department of Pharmaceutical Science and Technology, College of Chemistry and Biology, Donghua University, Shanghai, 201620, China.
  • Wang YH; Department of Pharmaceutical Science and Technology, College of Chemistry and Biology, Donghua University, Shanghai, 201620, China.
  • Qiu Y; Pudong New Area People's Hospital, Shanghai University of Medicine & Health Sciences, Shanghai, 201200, China. Electronic address: qiuyan2189@163.com.
  • Chen ZL; Department of Pharmaceutical Science and Technology, College of Chemistry and Biology, Donghua University, Shanghai, 201620, China. Electronic address: zlchen1967@qq.com.
Eur J Med Chem ; 181: 111553, 2019 Nov 01.
Article en En | MEDLINE | ID: mdl-31369932

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Bencimidazoles / Diseño de Fármacos / Receptor de Angiotensina Tipo 1 / Bloqueadores del Receptor Tipo 1 de Angiotensina II Límite: Animals Idioma: En Revista: Eur J Med Chem Año: 2019 Tipo del documento: Article País de afiliación: China Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Bencimidazoles / Diseño de Fármacos / Receptor de Angiotensina Tipo 1 / Bloqueadores del Receptor Tipo 1 de Angiotensina II Límite: Animals Idioma: En Revista: Eur J Med Chem Año: 2019 Tipo del documento: Article País de afiliación: China Pais de publicación: Francia