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N-Benzyl/Aryl Substituted Tryptanthrin as Dual Inhibitors of Indoleamine 2,3-Dioxygenase and Tryptophan 2,3-Dioxygenase.
Yang, Dan; Zhang, Shengnan; Fang, Xin; Guo, Leilei; Hu, Nan; Guo, Zhanling; Li, Xishuai; Yang, Shuangshuang; He, Jin Chao; Kuang, Chunxiang; Yang, Qing.
Afiliación
  • Yang D; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Zhang S; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Fang X; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Guo L; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Hu N; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Guo Z; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Li X; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Yang S; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • He JC; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
  • Kuang C; Department of Chemistry , Tongji University , Siping Road 1239 , Shanghai 200092 , China.
  • Yang Q; State Key Laboratory of Genetic Engineering, Department of Biochemistry, School of Life Sciences , Fudan University , Songhu Road 2005 , Shanghai 200438 , China.
J Med Chem ; 62(20): 9161-9174, 2019 10 24.
Article en En | MEDLINE | ID: mdl-31580660

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Quinazolinas / Triptófano Oxigenasa / Inhibidores Enzimáticos / Indolamina-Pirrol 2,3,-Dioxigenasa Límite: Animals / Female / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: China Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Quinazolinas / Triptófano Oxigenasa / Inhibidores Enzimáticos / Indolamina-Pirrol 2,3,-Dioxigenasa Límite: Animals / Female / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: China Pais de publicación: Estados Unidos