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Synthesis and Evaluation of 2-Aminothiophene Derivatives as Staphylococcus aureus Efflux Pump Inhibitors.
da Cruz, Rayssa M D; Zelli, Renaud; Benshain, Sarah; da Cruz, Ryldene M D; Siqueira-Júnior, José P; Décout, Jean-Luc; Mingeot-Leclercq, Marie-Paule; Mendonça-Junior, Francisco J B.
Afiliación
  • da Cruz RMD; Department of Biological Sciences, State University of Paraiba, Laboratory of Synthesis and Drug Delivery, João Pessoa, PB, Brazil.
  • Zelli R; Department of Pharmaceutical Sciences, Federal University of Paraiba, Post-Graduation Program in Natural and Synthetic Bioactive Products, João Pessoa, PB, Brazil.
  • Benshain S; Département de Pharmacochimie Moléculaire, University Grenoble Alpes, CNRS, Grenoble, France.
  • da Cruz RMD; Department of Pharmacologie Cellulaire et Moléculaire, Université Catholique de Louvain, Louvain Drug Research Institute, Brussels, Belgium.
  • Siqueira-Júnior JP; Département de Pharmacochimie Moléculaire, University Grenoble Alpes, CNRS, Grenoble, France.
  • Décout JL; Department of Pharmacologie Cellulaire et Moléculaire, Université Catholique de Louvain, Louvain Drug Research Institute, Brussels, Belgium.
  • Mingeot-Leclercq MP; Department of Pharmaceutical Sciences, Federal University of Paraiba, Post-Graduation Program in Natural and Synthetic Bioactive Products, João Pessoa, PB, Brazil.
  • Mendonça-Junior FJB; Department of Molecular Biology, Federal University of Paraiba, Laboratory of Microorganism Genetics, João Pessoa/PB, Brazil.
ChemMedChem ; 15(8): 716-725, 2020 04 20.
Article en En | MEDLINE | ID: mdl-32073756

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Staphylococcus aureus / Tiofenos / Proteínas Bacterianas / Proteínas Asociadas a Resistencia a Múltiples Medicamentos / Antibacterianos Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Brasil

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Staphylococcus aureus / Tiofenos / Proteínas Bacterianas / Proteínas Asociadas a Resistencia a Múltiples Medicamentos / Antibacterianos Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Brasil