MoS<sub>2</sub>-Calix[4]arene Catalyzed Synthesis and Molecular Docking Study of 2,4,5-Trisubstituted Imidazoles As Potent Inhibitors of <i>Mycobacterium tuberculosis</i>.

Raghu, Madihalli S; Pradeep Kumar, Chikkur B; Prasad, Kodalapura N Nagendra; Prashanth, Maralekere K; Kumarswamy, Yogesh K; Chandrasekhar, Sunkara; Veeresh, Bantal

MoS₂-Calix[4]arene Catalyzed Synthesis and Molecular Docking Study of 2,4,5-Trisubstituted Imidazoles As Potent Inhibitors of Mycobacterium tuberculosis.

Raghu, Madihalli S; Pradeep Kumar, Chikkur B; Prasad, Kodalapura N Nagendra; Prashanth, Maralekere K; Kumarswamy, Yogesh K; Chandrasekhar, Sunkara; Veeresh, Bantal.

Afiliación

Raghu MS; Department of Chemistry, New Horizon College of Engineering, Bangalore 560 103, India.
Pradeep Kumar CB; Department of Chemistry, Malnad College of Engineering, Hassan 573 202, India.
Prasad KNN; Department of Physics, B N M Institute of Technology, Bangalore 560 070, India.
Prashanth MK; Department of Chemistry, B N M Institute of Technology, Bangalore 560 070, India.
Kumarswamy YK; Department of Chemistry, School of Engineering and Technology, Jain University, Ramanagara, 562 112, India.
Chandrasekhar S; Department of Physics, B N M Institute of Technology, Bangalore 560 070, India.
Veeresh B; Department of Pharmacology, G. Pullareddy College of Pharmacy, Mehdipatnam, Hyderabad 580 028, India.

ACS Comb Sci ; 22(10): 509-518, 2020 10 12.

Article en En | MEDLINE | ID: mdl-32806898

Asunto(s)

3-Oxoacil-(Proteína Transportadora de Acil) Reductasa/antagonistas & inhibidores; Antituberculosos/síntesis química; Proteínas Bacterianas/antagonistas & inhibidores; Calixarenos/química; Disulfuros/química; Inhibidores Enzimáticos/síntesis química; Imidazoles/síntesis química; Molibdeno/química; Mycobacterium tuberculosis/efectos de los fármacos; Fenoles/química; Animales; Antituberculosos/farmacología; Catálisis; Chlorocebus aethiops; Evaluación Preclínica de Medicamentos; Inhibidores Enzimáticos/farmacología; Humanos; Imidazoles/farmacología; Pruebas de Sensibilidad Microbiana; Simulación del Acoplamiento Molecular; Unión Proteica; Bibliotecas de Moléculas Pequeñas; Relación Estructura-Actividad; Células Vero/efectos de los fármacos

Palabras clave

MoS2-supported-calix[4]arene (MoS2-CA4); Mycobacterium tuberculosis; docking study; imidazoles; nanoparticles

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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Fenoles / Proteínas Bacterianas / Calixarenos / Disulfuros / Inhibidores Enzimáticos / 3-Oxoacil-(Proteína Transportadora de Acil) Reductasa / Imidazoles / Molibdeno / Mycobacterium tuberculosis / Antituberculosos Límite: Animals / Humans Idioma: En Revista: ACS Comb Sci Año: 2020 Tipo del documento: Article País de afiliación: India Pais de publicación: Estados Unidos

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