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Design, synthesis and biological evaluation of imidazole and triazole-based carbamates as novel aromatase inhibitors.
Ammazzalorso, Alessandra; Gallorini, Marialucia; Fantacuzzi, Marialuigia; Gambacorta, Nicola; De Filippis, Barbara; Giampietro, Letizia; Maccallini, Cristina; Nicolotti, Orazio; Cataldi, Amelia; Amoroso, Rosa.
Afiliación
  • Ammazzalorso A; Unit of Medicinal Chemistry, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy. Electronic address: alessandra.ammazzalorso@unich.it.
  • Gallorini M; Unit of Anatomy, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy.
  • Fantacuzzi M; Unit of Medicinal Chemistry, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy.
  • Gambacorta N; Unit of Medicinal Chemistry, Department of Farmacia-Scienze Del Farmaco, "A. Moro" University, Bari, Italy.
  • De Filippis B; Unit of Medicinal Chemistry, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy.
  • Giampietro L; Unit of Medicinal Chemistry, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy.
  • Maccallini C; Unit of Medicinal Chemistry, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy.
  • Nicolotti O; Unit of Medicinal Chemistry, Department of Farmacia-Scienze Del Farmaco, "A. Moro" University, Bari, Italy.
  • Cataldi A; Unit of Anatomy, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy.
  • Amoroso R; Unit of Medicinal Chemistry, Department of Pharmacy, "G. D'Annunzio" University, Chieti, Italy.
Eur J Med Chem ; 211: 113115, 2021 Feb 05.
Article en En | MEDLINE | ID: mdl-33360796

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Triazoles / Carbamatos / Inhibidores de la Aromatasa / Imidazoles Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2021 Tipo del documento: Article Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Triazoles / Carbamatos / Inhibidores de la Aromatasa / Imidazoles Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2021 Tipo del documento: Article Pais de publicación: Francia