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Evaluation and docking of indole sulfonamide as a potent inhibitor of α-glucosidase enzyme in streptozotocin -induced diabetic albino wistar rats.
Taha, Muhammad; Imran, Syahrul; Salahuddin, Mohammed; Iqbal, Naveed; Rahim, Fazal; Uddin, Nizam; Shehzad, Adeeb; Khalid Farooq, Rai; Alomari, Munther; Mohammed Khan, Khalid.
Afiliación
  • Taha M; Department of Clinical Pharmacy Research, Institute for Research and Medical Consultations (IRMC), Imam Abdulrahman Bin Faisal University, P.O. Box 31441, Dammam, Saudi Arabia. Electronic address: mtaha@iau.edu.sa.
  • Imran S; Atta-ur-Rahman Institute for Natural Product Discovery, Universiti Teknologi MARA (UiTM), Puncak Alam Campus, 42300 Bandar Puncak Alam, Selangor, Malaysia.
  • Salahuddin M; Department of Clinical Pharmacy Research, Institute for Research and Medical Consultations (IRMC), Imam Abdulrahman Bin Faisal University, P.O. Box 31441, Dammam, Saudi Arabia.
  • Iqbal N; Department of Chemistry University of Poonch, Rawalakot, AJK, Pakistan.
  • Rahim F; Department of Chemistry, Hazara University, Mansehra 21300, Khyber Pakhtunkhwa, Pakistan.
  • Uddin N; Department of Chemistry, University of Karachi, Karachi 75270, Pakistan.
  • Shehzad A; Department of Clinical Pharmacy Research, Institute for Research and Medical Consultations (IRMC), Imam Abdulrahman Bin Faisal University, P.O. Box 31441, Dammam, Saudi Arabia.
  • Khalid Farooq R; Department of Neuroscience Research, Institute for Research and Medical Consultations (IRMC), Imam Abdulrahman Bin Faisal University, P.O. Box 1982, Dammam 31441, Saudi Arabia.
  • Alomari M; Department of Stem Cell Biology, Institute for Research and Medical Consultations (IRMC), Imam Abdulrahman Bin Faisal University, P.O. Box 1982, Dammam 31441, Saudi Arabia.
  • Mohammed Khan K; H. E. J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi 75270, Pakistan.
Bioorg Chem ; 110: 104808, 2021 05.
Article en En | MEDLINE | ID: mdl-33756236

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Sulfonamidas / Diabetes Mellitus Experimental / Alfa-Glucosidasas / Simulación del Acoplamiento Molecular / Inhibidores de Glicósido Hidrolasas / Hipoglucemiantes / Indoles Límite: Animals Idioma: En Revista: Bioorg Chem Año: 2021 Tipo del documento: Article Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Sulfonamidas / Diabetes Mellitus Experimental / Alfa-Glucosidasas / Simulación del Acoplamiento Molecular / Inhibidores de Glicósido Hidrolasas / Hipoglucemiantes / Indoles Límite: Animals Idioma: En Revista: Bioorg Chem Año: 2021 Tipo del documento: Article Pais de publicación: Estados Unidos