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Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists.
Jiang, Shan; Iliopoulos-Tsoutsouvas, Christos; Tong, Fei; Brust, Christina A; Keenan, Catherine M; Raghav, Jimit Girish; Hua, Tian; Wu, Simiao; Ho, Jo-Hao; Wu, Yiran; Grim, Travis W; Zvonok, Nikolai; Thakur, Ganesh A; Liu, Zhi-Jie; Sharkey, Keith A; Bohn, Laura M; Nikas, Spyros P; Makriyannis, Alexandros.
Afiliación
  • Brust CA; Department of Molecular Medicine, The Scripps Research Institute, Jupiter, Florida 33458, United States.
  • Keenan CM; Hotchkiss Brain Institute and Snyder Institute for Chronic Diseases, Department of Physiology and Pharmacology, University of Calgary, Calgary, Alberta T2N 4N1, Canada.
  • Hua T; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Ho JH; Department of Molecular Medicine, The Scripps Research Institute, Jupiter, Florida 33458, United States.
  • Wu Y; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Grim TW; Department of Molecular Medicine, The Scripps Research Institute, Jupiter, Florida 33458, United States.
  • Liu ZJ; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Sharkey KA; Hotchkiss Brain Institute and Snyder Institute for Chronic Diseases, Department of Physiology and Pharmacology, University of Calgary, Calgary, Alberta T2N 4N1, Canada.
  • Bohn LM; Department of Molecular Medicine, The Scripps Research Institute, Jupiter, Florida 33458, United States.
J Med Chem ; 64(7): 3870-3884, 2021 04 08.
Article en En | MEDLINE | ID: mdl-33761251

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Cannabinoides / Receptor Cannabinoide CB1 / Receptor Cannabinoide CB2 / Agonistas de Receptores de Cannabinoides Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2021 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Cannabinoides / Receptor Cannabinoide CB1 / Receptor Cannabinoide CB2 / Agonistas de Receptores de Cannabinoides Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2021 Tipo del documento: Article