Conformational-Design-Driven Discovery of EZM0414: A Selective, Potent SETD2 Inhibitor for Clinical Studies.

Alford, Joshua S; Lampe, John W; Brach, Dorothy; Chesworth, Richard; Cosmopoulos, Kat; Duncan, Kenneth W; Eckley, Sean T; Kutok, Jeffrey L; Raimondi, Alejandra; Riera, Thomas V; Shook, Brian; Tang, Cuyue; Totman, Jennifer; Farrow, Neil A

Alford, Joshua S; Lampe, John W; Brach, Dorothy; Chesworth, Richard; Cosmopoulos, Kat; Duncan, Kenneth W; Eckley, Sean T; Kutok, Jeffrey L; Raimondi, Alejandra; Riera, Thomas V; Shook, Brian; Tang, Cuyue; Totman, Jennifer; Farrow, Neil A.

Afiliación

Alford JS; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Lampe JW; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Brach D; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Chesworth R; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Cosmopoulos K; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Duncan KW; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Eckley ST; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Kutok JL; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Raimondi A; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Riera TV; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Shook B; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Tang C; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Totman J; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.
Farrow NA; Epizyme Inc., 50 Hampshire Street, Sixth Floor, Cambridge, Massachusetts 02139, United States.

ACS Med Chem Lett ; 13(7): 1137-1143, 2022 Jul 14.

Article en En | MEDLINE | ID: mdl-35859865

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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2022 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

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