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Synthesis and biological evaluation of coumarin-thiazole hybrids as selective carbonic anhydrase IX and XII inhibitors.
Thacker, Pavitra S; Newaskar, Vaishnavi; Angeli, Andrea; Sigalapalli, Dilep Kumar; Goud, Nerella Sridhar; Chirra, Hepsibha; Shaik, Afzal B; Arifuddin, Mohammed; Supuran, Claudiu T.
Afiliación
  • Thacker PS; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
  • Newaskar V; Department of Pharmaceutical Chemistry, L.J. Institute of Pharmacy, L.J. University, Ahmedabad, Gujarat, India.
  • Angeli A; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
  • Sigalapalli DK; Neurofarba Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, Università degl iStudi di Firenze, Florence, Italy.
  • Goud NS; Department of Pharmaceutical Chemistry, Vignan Pharmacy College, Jawaharlal Nehru Technological University, Guntur, Andhra Pradesh, India.
  • Chirra H; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
  • Shaik AB; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
  • Arifuddin M; Department of Pharmaceutical Chemistry, Vignan Pharmacy College, Jawaharlal Nehru Technological University, Guntur, Andhra Pradesh, India.
  • Supuran CT; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
Arch Pharm (Weinheim) ; 355(12): e2200232, 2022 Dec.
Article en En | MEDLINE | ID: mdl-36122182

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores de Anhidrasa Carbónica / Anhidrasas Carbónicas Límite: Humans Idioma: En Revista: Arch Pharm (Weinheim) Año: 2022 Tipo del documento: Article País de afiliación: India Pais de publicación: Alemania

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores de Anhidrasa Carbónica / Anhidrasas Carbónicas Límite: Humans Idioma: En Revista: Arch Pharm (Weinheim) Año: 2022 Tipo del documento: Article País de afiliación: India Pais de publicación: Alemania