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3-Substituted-2,3-Dihydrothiazole as a promising scaffold to design EGFR inhibitors.
El-Haggar, Radwan; Hammad, Sherif F; Alsantali, Reem I; Alrooqi, Munira M; El Hassab, Mahmoud A; Masurier, Nicolas; Ahmed, Marwa F.
Afiliación
  • El-Haggar R; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Ain Helwan 11795, Cairo, Egypt; Institut des Biomolécules Max Mousseron (IBMM), UMR 5247, CNRS, Université de Montpellier, ENSCM, 34293 Montpellier, France. Electronic address: radwan_elhaggar@pharm.helwan.edu.eg.
  • Hammad SF; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Ain Helwan 11795, Cairo, Egypt; Basic and Applied Science Institute, Egypt-Japan University of Science and Technology (E-JUST), New Borg El-Arab City 21934, Alexandria, Egypt.
  • Alsantali RI; Department of Pharmaceutical Chemistry, College of Pharmacy, Taif University, P.O. Box 11099, Taif 21944, Saudi Arabia.
  • Alrooqi MM; Department of Chemistry, Faculty of Applies Science, Umm Al-Qura University, 21944, Makkah, Saudi Arabia.
  • El Hassab MA; Department of Medicinal Chemistry, Faculty of Pharmacy, King Salman International University (KSIU), South Sinai, Egypt.
  • Masurier N; Institut des Biomolécules Max Mousseron (IBMM), UMR 5247, CNRS, Université de Montpellier, ENSCM, 34293 Montpellier, France. Electronic address: nicolas.masurier@umontpellier.fr.
  • Ahmed MF; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Ain Helwan 11795, Cairo, Egypt; Department of Pharmaceutical Chemistry, College of Pharmacy, Taif University, P.O. Box 11099, Taif 21944, Saudi Arabia. Electronic address: marwa_farag@pharm.helwan.edu.eg.
Bioorg Chem ; 129: 106172, 2022 Dec.
Article en En | MEDLINE | ID: mdl-36182865

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores de Proteínas Quinasas / Antineoplásicos Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Bioorg Chem Año: 2022 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores de Proteínas Quinasas / Antineoplásicos Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Bioorg Chem Año: 2022 Tipo del documento: Article