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Discovery of a brain-sparing GIRK1/4 inhibitor for pharmacological cardioversion of atrial fibrillation.
Peukert, Stefan; Gulgeze Efthymiou, Hatice Belgin; Mo, Ruowei; Peng, Yunshan; Ma, Fupeng; Barbe, Guillaume; Bebernitz, Gregory; Fridrich, Cary; Buono, Chiara; Williams, Eric T; Daniels, Thomas; Li, Lisha; Zhang, Xia; Adachi, Yuichiro; Abe, Mie; Taggart, Andrew K P.
Afiliación
  • Peukert S; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA. Electronic address: stefan.peukert@novartis.com.
  • Gulgeze Efthymiou HB; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Mo R; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Peng Y; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Ma F; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Barbe G; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Bebernitz G; Former Novartis Employee, USA.
  • Fridrich C; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Buono C; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Williams ET; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Daniels T; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Li L; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Zhang X; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Adachi Y; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
  • Abe M; Former Novartis Employee, USA.
  • Taggart AKP; Novartis Institutes for Biomedical Research, 181 Massachusetts Avenue, Cambridge, MA 02139, USA.
Bioorg Med Chem Lett ; 85: 129237, 2023 04 01.
Article en En | MEDLINE | ID: mdl-36924945

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Fibrilación Atrial Tipo de estudio: Risk_factors_studies Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Fibrilación Atrial Tipo de estudio: Risk_factors_studies Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article Pais de publicación: Reino Unido